SCHEMBL12470256

SCHEMBL12470256

CCOc1ccc2c(c1)OC(C)(C)CC21C(=O)N(Cc2ccc(OC)cc2)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 10/20 0.51
L3MBTL1 Q9Y468 1/20 0.42
OPRL1 P41146 1/20 0.42
MAPT P10636 2/20 0.41
LMNA P02545 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
CYP3A4 P08684 1/20 0.40
MMP12 P39900 1/20 0.40
ADAMTS5 Q9UNA0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12469858 0.92 SCN9A (0.45) SCN9AMAPTLMNACYP3A4
SCHEMBL12470231 0.90 MAOB (0.46) SCN9AMAPTCYP3A4
SCHEMBL12470286 0.90 SCN9A (0.43) SCN9AMAPTCYP3A4
SCHEMBL12470330 0.87 MAOB (0.47) SCN9AMAPTCYP3A4
SCHEMBL12471313 0.86 SCN9A (0.47) SCN9AL3MBTL1MAPTCYP3A4
SCHEMBL12470315 0.85 MAPT (0.42) SCN9AMAPTCYP3A4
SCHEMBL12470852 0.85 SCN9A (0.42) SCN9AMAPTPTGDR2
SCHEMBL12470309 0.84 SCN9A (0.45) SCN9AMAPTCYP3A4
SCHEMBL12470044 0.84 SCN9A (0.44) SCN9ACYP3A4
SCHEMBL12470080 0.83 SCN9A (0.47) SCN9AMAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012049555-A1 SPIROCYCLIC COMPOUNDS AS VOLTAGE-GATED SODIUM CHANNEL MODULATORS LUPIN LIMITED (IN) 2012-04-19 WO disclosed