SCHEMBL12484207

SCHEMBL12484207

CCOC(=O)c1sc(-c2ccc(F)c(Cl)c2)c(C)c1-c1ccc(S(N)(=O)=O)cc1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 9/20 0.59
PTGS1 P23219 7/20 0.46
PTGS2 P35354 7/20 0.46
CA2 P00918 3/20 0.41
CA1 P00915 2/20 0.41
CA9 Q16790 2/20 0.41
CA12 O43570 1/20 0.41
CA4 P22748 1/20 0.41
SOS1 Q07889 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12484020 0.91 CHRNA7 (0.57) CHRNA7PTGS1PTGS2CA2CA1
SCHEMBL12483079 0.91 CHRNA7 (0.60) CHRNA7PTGS1PTGS2CA2CA1
SCHEMBL12483720 0.88 CHRNA7 (0.77) CHRNA7PTGS1PTGS2CA2SOS1
SCHEMBL12483675 0.88 CHRNA7 (0.76) CHRNA7PTGS1PTGS2CA2CA1
SCHEMBL12482858 0.87 CHRNA7 (0.56) CHRNA7PTGS1PTGS2CA2CA1
SCHEMBL12483588 0.87 CHRNA7 (0.60) CHRNA7CA2CA1CA9CA12
SCHEMBL12483956 0.87 CHRNA7 (0.59) CHRNA7PTGS1PTGS2CA2SOS1
SCHEMBL12483144 0.86 CHRNA7 (0.60) CHRNA7PTGS1PTGS2CA2CA1
SCHEMBL12484141 0.85 CHRNA7 (0.53) CHRNA7PTGS1PTGS2CA2CA1
SCHEMBL12483858 0.84 CHRNA7 (0.59) CHRNA7PTGS1PTGS2CA2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2678327-A1 HETEROARYL DERIVATIVES AS ALPHA7 NACHR MODULATORS Lupin Limited (IN) 2014-01-01 EP disclosed
WO-2012114285-A9 HETEROARYL DERIVATIVES AS ALPHA7 NACHR MODULATORS LUPIN LIMITED (IN) 2012-10-18 WO disclosed
WO-2012114285-A1 HETEROARYL DERIVATIVES AS ALPHA7 NACHR MODULATORS LUPIN LIMITED (IN) 2012-08-30 WO disclosed