SCHEMBL12487181

SCHEMBL12487181

CN1CCN(c2ncnc(Nc3cccc(CS(N)(=O)=O)c3)n2)CC1.NS(=O)(=O)Cc1cccc(Nc2ncnc(N3CCNCC3)n2)c1.NS(=O)(=O)Cc1cccc(Nc2ncnc(N3CCOCC3)n2)c1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
POLB P06746 2/20 0.47
CA12 O43570 2/20 0.45
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA9 Q16790 2/20 0.45
SCN9A Q15858 10/20 0.45
CCNT1 O60563 1/20 0.44
CCNE2 O96020 1/20 0.44
CCNE1 P24864 1/20 0.44
CDK2 P24941 1/20 0.44
CDK9 P50750 1/20 0.44
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
FGFR3 P22607 2/20 0.42
KDR P35968 2/20 0.42
BMPR2 Q13873 1/20 0.42
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12486174 0.89 SCN9A (0.53) SCN9ACCNT1CCNE2CCNE1CDK2
SCHEMBL12486402 0.89 CCNT1 (0.49) POLBSCN9ACCNT1CCNE2CCNE1
SCHEMBL12485723 0.89 CA12 (0.52) POLBCA12CA1CA2CA9
SCHEMBL12487189 0.88 USP2 (0.49) USP2SMN1; SMN2POLBCA12CA1
SCHEMBL12485572 0.81 CCNT1 (0.54) SMN1; SMN2SCN9ACCNT1CCNE2CCNE1
SCHEMBL12487113 0.80 CDK2 (0.53) SMN1; SMN2SCN9ACCNT1CCNE2CCNE1
SCHEMBL12486627 0.77 CCNT1 (0.50) SCN9ACCNT1CCNE2CCNE1CDK2
SCHEMBL12487046 0.75 CCNT1 (0.43) SCN9ACCNT1CCNE2CCNE1CDK2
SCHEMBL12486620 0.75 SCN9A (0.67) SCN9A
SCHEMBL12487169 0.74 SCN9A (0.51) SCN9ACCNT1CCNE2CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2680852-A1 PHARMACEUTICALLY ACTIVE DISUBSTITUTED TRIAZINE DERIVATIVES Lead Discovery Center GmbH (DE) 2014-01-08 EP claimed
WO-2012117048-A1 PHARMACEUTICALLY ACTIVE DISUBSTITUTED TRIAZINE DERIVATIVES LEAD DISCOVERY CENTER GMBH (DE) 2012-09-07 WO claimed