SCHEMBL12499504

SCHEMBL12499504

CCOC(=O)C1C(c2ccccc2)C1c1ccc(N)c(Br)c1

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
PPARG P37231 4/20 0.44
FABP7 O15540 3/20 0.44
FABP5 Q01469 2/20 0.44
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
GAA P10253 1/20 0.44
TP53 P04637 2/20 0.44
POLB P06746 1/20 0.42
HDAC4 P56524 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15768958 1.00 TSHR (0.45) TSHRPPARGFABP7FABP5MEN1
SCHEMBL15783747 0.84 FABP7 (0.60) TSHRPPARGFABP7FABP5MEN1
SCHEMBL14276798 0.83 TSHR (0.60) TSHRPPARGFABP7FABP5MEN1
SCHEMBL5122894 0.83 TSHR (0.60) TSHRPPARGFABP7FABP5MEN1
SCHEMBL15768614 0.83 HDAC4 (0.59) TSHRPPARGFABP7FABP5MEN1
SCHEMBL15768992 0.82 TSHR (0.53) TSHRPPARGFABP7FABP5MEN1
SCHEMBL12498187 0.82 GAA (0.42) TSHRPPARGFABP7FABP5MEN1
SCHEMBL12694435 0.82 GAA (0.42) TSHRPPARGFABP7FABP5MEN1
SCHEMBL15768581 0.81 HDAC4 (0.61) TSHRPPARGFABP7FABP5MEN1
SCHEMBL18462855 0.80 GAA (0.63) TSHRPPARGFABP7FABP5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2667709-A1 HISTONE DEACETYLASE INHIBITORS AND COMPOSITIONS AND METHODS OF USE THEREOF CHDI Foundation, Inc. (US) 2013-12-04 EP disclosed
WO-2012103008-A1 HISTONE DEACETYLASE INHIBITORS AND COMPOSITIONS AND METHODS OF USE THEREOF CHDI FOUNDATION, INC. (US) 2012-08-02 WO disclosed