SCHEMBL12502136

SCHEMBL12502136

CC1(C)CN(c2nc(Cl)nc3c2CCC3c2ccc(F)cc2)CCO1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 1/20 0.36
FFAR2 O15552 9/20 0.36
PDE10A Q9Y233 1/20 0.35
ACACB O00763 1/20 0.32
PIK3CA P42336 1/20 0.31
MTOR P42345 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
LRRK2 Q5S007 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL512835 0.82 HRH3 (0.34) HRH4HRH3
SCHEMBL511681 0.81 HRH3 (0.32) HRH4HRH3
SCHEMBL18559820 0.81 HRH3 (0.41) PDE10AHRH4HRH3
SCHEMBL511790 0.81 HRH3 (0.35) PDE10AHRH4HRH3
SCHEMBL512628 0.81 CYP3A4 (0.34) HRH4HRH3
SCHEMBL513595 0.80 SMN1; SMN2 (0.43) HRH4HRH3
SCHEMBL512509 0.80 CYP3A4 (0.30)
SCHEMBL511704 0.79 MAOB (0.36) FFAR2PDE10AHRH4HRH3
SCHEMBL18559791 0.79 CYP3A4 (0.33) HRH4HRH3
SCHEMBL512280 0.78 GAK (0.38) FFAR2HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2668168-A1 COMPOUNDS FOR THE REDUCTION OF ß-AMYLOID PRODUCTION Bristol-Myers Squibb Company (US) 2013-12-04 EP disclosed
WO-2012103297-A1 COMPOUNDS FOR THE REDUCTION OF β-AMYLOID PRODUCTION BRISTOL-MYERS SQUIBB COMPANY (US) 2012-08-02 WO disclosed