SCHEMBL1250846

SCHEMBL1250846

O=C(NC1CCNC1)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
HDAC4 P56524 1/20 0.52
KDM1A O60341 1/20 0.51
KDR P35968 1/20 0.50
ACSS2 Q9NR19 1/20 0.48
MAPK1 P28482 1/20 0.48
OPRK1 P41145 1/20 0.48
CTSL P07711 1/20 0.48
CTSB P07858 1/20 0.48
CTSK P43235 1/20 0.48
EZH2 Q15910 1/20 0.48
SMYD3 Q9H7B4 1/20 0.48
PARP1 P09874 1/20 0.47
CARM1 Q86X55 1/20 0.47
PRMT6 Q96LA8 1/20 0.47
GRM5 P41594 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230051 1.00 MEN1 (0.54) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL8491815 1.00 MEN1 (0.54) MEN1KMT2ANPC1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL28156652 0.98 MEN1 (0.53) MEN1KMT2ANPC1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL994487 0.98 MEN1 (0.53) MEN1KMT2ANPC1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL28155972 0.98 MEN1 (0.53) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL23638927 0.91 NPC1 (0.69) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL1163022 0.90 MAPK1 (0.59) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL1163023 0.90 MAPK1 (0.59) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL28280152 0.90 MAPK1 (0.59) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL594567 0.90 NPC1 (0.62) MEN1KMT2ANPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 61 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023046117-A1 FGFR INHIBITORS AND METHODS OF USE THEREOF 3H PHARMACEUTICALS CO., LTD. (CN) 2023-03-30 WO claimed
EP-3612174-B1 METHODS AND PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF DISEASES ASSOCIATED WITH REDUCED CFTR FUNCTION INST NAT SANTE RECH MED (FR) 2023-02-22 EP claimed
US-9382197-B2 Substituted hydroxamic acids and uses thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2016-07-05 US claimed
EP-1188744-B1 Process for producing optically active 1H-3-aminopyrrolidine and derivatives thereof MITSUBISHI CHEM CORP (JP) 2005-11-02 EP claimed
US-5686482-A DOPAMINE RECEPTOR ANTAGONIST YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1997-11-11 US claimed
CN-1147248-A N- (3-pyrrolidinyl) benzamide derivatives YAMANOUCHI PHARMA CO LTD (JP) 1997-04-09 CN claimed
EP-0757985-A1 N-(3-PYRROLIDINYL)BENZAMIDE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1997-02-12 EP claimed
US-4049821-A 3-AMINO-PYRROLIDINYL-BENZAMIDE A. H. ROBINS COMPANY, INC. (US) 1977-09-20 US claimed
CN-118239926-A TLR7 and 8 inhibitors, preparation method and application thereof 上海深势唯思科技有限责任公司 2024-06-25 CN disclosed
US-20240083844-A1 KINASE INHIBITORS AND USES THEREOF ABM THERAPEUTICS CORPORATION (US) 2024-03-14 US disclosed
EP-4157888-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS Cullgen (Shanghai), Inc. (CN) 2023-04-05 EP disclosed
WO-2023046117-A1 FGFR INHIBITORS AND METHODS OF USE THEREOF 3H PHARMACEUTICALS CO., LTD. (CN) 2023-03-30 WO disclosed
WO-2022262854-A1 CLY SERIES COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN PREPARATION OF DRUGS 南京韦尔优众医药有限公司 2022-12-22 WO disclosed
WO-2021239117-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS CULLGEN (SHANGHAI) , INC. (CN) 2021-12-02 WO disclosed
US-4073796-A ANTIEMETIC A. H. ROBINS COMPANY, INC. (US) 1978-02-14 US disclosed
US-4049821-A 3-AMINO-PYRROLIDINYL-BENZAMIDE A. H. ROBINS COMPANY, INC. (US) 1977-09-20 US disclosed
US-4039678-A N-(SUBSTITUTED-3-PYRROLIDINYL)-1-NAPHTHALENE CARBOXAMIDES A. H. ROBINS COMPANY, INCORPORATED (US) 1977-08-02 US disclosed
US-4002757-A ANTIEMETIC AGENTS A. H. ROBINS COMPANY, INCORPORATED (US) 1977-01-11 US disclosed
US-3966957-A Method for controlling emesis with N-(1-substituted-3-pyrrolidinyl)benzamides and thiobenzamides A. H. ROBINS COMPANY, INCORPORATED (US) 1976-06-29 US disclosed
US-3963745-A Method for controlling emesis with N-(1-substituted-3-pyrrolidinyl)benzamides and thiobenzamides A. H. ROBINS COMPANY, INCORPORATED (US) 1976-06-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240083844-A1 KINASE INHIBITORS AND USES THEREOF MINK1, PTK2, PLK4 MEN1 505/4885KMT2A 633/4885NPC1 4603/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.