SCHEMBL12510600

SCHEMBL12510600

BNc1cccc(Nc2cc(Cl)ncn2)c1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.51
EGFR P00533 9/20 0.48
ERBB3 P21860 3/20 0.47
MKNK1 Q9BUB5 1/20 0.46
TNNI3K Q59H18 5/20 0.43
MEN1 O00255 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
THRB P10828 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3952295 0.83 EGFR (0.66) NPC1EGFRERBB3MKNK1TNNI3K
Hydrochloric Acid SCHEMBL2173883 0.82 EGFR (0.64) NPC1EGFRERBB3MKNK1TNNI3K
SCHEMBL857502 0.81 NPC1 (0.63) NPC1EGFRERBB3MKNK1TNNI3K
SCHEMBL2279563 0.81 MEN1 (0.56) NPC1EGFRERBB3MKNK1MEN1
SCHEMBL691533 0.81 EGFR (0.57) NPC1EGFRERBB3TNNI3K
SCHEMBL2279629 0.81 EGFR (0.59) NPC1EGFRERBB3MKNK1TNNI3K
SCHEMBL20093470 0.81 NPC1 (0.51) NPC1EGFRERBB3MKNK1TNNI3K
SCHEMBL657571 0.81 TP53 (0.62) NPC1EGFRERBB3MKNK1TP53
Hydrochloric Acid SCHEMBL2176643 0.80 NPC1 (0.61) NPC1EGFRERBB3MKNK1TNNI3K
SCHEMBL1243031 0.79 EGFR (0.51) NPC1EGFRERBB3MKNK1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7982036-B2 4,6-disubstitued pyrimidines useful as kinase inhibitors AVILA THERAPEUTICS, INC. (US) 2011-07-19 US disclosed
US-20090137588-A1 HETEROARYL COMPOUNDS AND USES THEREOF AVILA THERAPEUTICS, INC. (US) 2009-05-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090137588-A1 HETEROARYL COMPOUNDS AND USES THEREOF ABCG2, CYP3A43, CYP3A5 NPC1 48/4885EGFR 1981/4885ERBB3 294/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.