SCHEMBL1256451

SCHEMBL1256451

c1ccc(Sc2ccco2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.38
MAPT P10636 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
MGLL Q99685 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MAOA P21397 2/20 0.35
MAOB P27338 2/20 0.35
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
ALDH1A1 P00352 4/20 0.33
MAPK1 P28482 2/20 0.33
KDM4E B2RXH2 1/20 0.33
PKM P14618 1/20 0.33
NTSR1 P30989 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25498805 0.82
SCHEMBL2209772 0.82 TP53 (0.41) HPGDMAPTHSD17B10NPC1RAB9A
SCHEMBL9087579 0.77 MAP2K2 (0.41) HPGDMAPTSMN1; SMN2HSD17B10CYP1A2
SCHEMBL24359523 0.71 TDP1 (0.32) MAPTSMN1; SMN2HSD17B10CYP3A4ALDH1A1
SCHEMBL2212333 0.71 TP53 (0.41) HPGDMAPTHSD17B10NPC1RAB9A
Diphenylsulfane SCHEMBL28332331 0.69 HPGD (0.60) HPGDMAPTSMN1; SMN2MGLLHSD17B10
Diphenylsulfane SCHEMBL452 0.69 HPGD (0.60) HPGDMAPTSMN1; SMN2MGLLHSD17B10
Diphenylsulfane SCHEMBL27611905 0.69 HPGD (0.60) HPGDMAPTSMN1; SMN2MGLLHSD17B10
Diphenylsulfane SCHEMBL27714827 0.69 HPGD (0.60) HPGDMAPTSMN1; SMN2MGLLHSD17B10
Diphenylsulfane SCHEMBL7109540 0.69 HPGD (0.60) HPGDMAPTSMN1; SMN2MGLLHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119039573-A Conjugated polymer based on fluorine-containing acenaphthoquinoxaline condensed ring unit, and preparation method and application thereof 广东工业大学 2024-11-29 CN disclosed
US-9604316-B2 Tin-based solder composition with low void characteristic GLOBALFOUNDRIES INC. (KY) 2017-03-28 US disclosed
US-9465290-B2 Near-infrared absorbing film compositions GLOBALFOUNDRIES INC. (KY) 2016-10-11 US disclosed
US-9348228-B2 Acid-strippable silicon-containing antireflective coating GLOBALFOUNDRIES INC. (KY) 2016-05-24 US disclosed
US-20160082551-A1 TIN-BASED SOLDER COMPOSITION WITH LOW VOID CHARACTERISTIC GLOBALFOUNDRIES U.S. INC. 2016-03-24 US disclosed
US-20140210034-A1 NEAR-INFRARED ABSORBING FILM COMPOSITIONS INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2014-07-31 US disclosed
WO-2014107476-A1 ACID-STRIPPABLE SILICON-CONTAINING ANTIREFLECTIVE COATING INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2014-07-10 WO disclosed
US-8772376-B2 Near-infrared absorbing film compositions INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2014-07-08 US disclosed
US-20140186774-A1 ACID-STRIPPABLE SILICON-CONTAINING ANTIREFLECTIVE COATING INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2014-07-03 US disclosed
US-8586283-B2 Near-infrared absorbing film compositions INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2013-11-19 US disclosed
US-5594021-A VASOCONSTRICTORS TEXAS BIOTECHNOLOGY CORPORATION (US) 1997-01-14 US disclosed
US-5571821-A CARDIOVASCULAR DISORDERS TO MODULATE ENDOTHELIN, HYPOTENSIVE AGENTS AND VASOCONSTRICTION TEXAS BIOTECHNOLOGY CORPORATION (US) 1996-11-05 US disclosed
WO-1996031492-A1 THIENYL-, FURYL-, PYRROLYL- AND BIPHENYLSULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN TEXAS BIOTECHNOLOGY CORPORATION (US) 1996-10-10 WO disclosed
EP-0699191-A1 SULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN TEXAS BIOTECHNOLOGY CORPORATION (US) 1996-03-06 EP disclosed
US-5389673-A HYPOGLYCEMIC AGENTS; ANTICHOLESTEROL AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1995-02-14 US disclosed
US-5389672-A ANTICHOLESTEROL AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1995-02-14 US disclosed
US-5389671-A ANTIULCER AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1995-02-14 US disclosed
WO-1994027979-A1 SULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN IMMUNOPHARMACEUTICS, INC. (US) 1994-12-08 WO disclosed
US-5314913-A Anticholesterol, antiulcer AMERICAN HOME PRODUCTS CORPORATION (US) 1994-05-24 US disclosed
US-4294838-A ANTIBRONCHOSPASMOLYTIC AGENTS WARNER-LAMBERT COMPANY, A CORP. OF DE 1981-10-13 US disclosed