SCHEMBL12572304

SCHEMBL12572304

C=S(=O)(N[C@H]1CC[C@H](C(=O)N[C@H](C)c2ccc(F)cc2)CC1)c1ccc(-c2cnn(C)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KIT P10721 14/20 0.50
GPR55 Q9Y2T6 1/20 0.44
MAPK1 P28482 1/20 0.41
ACACB O00763 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12551248 0.91 KIT (0.51) KITGPR55MAPK1ACACB
SCHEMBL12572232 0.84 KIT (0.44) KITACACB
SCHEMBL12551042 0.83 KIT (0.49) KITGPR55MAPK1ACACB
SCHEMBL256333 0.82 ACACB (0.57) KITACACB
SCHEMBL16622564 0.82 KIT (0.55) KITGPR55
SCHEMBL12551291 0.78 KIT (0.46) KITACACB
SCHEMBL1953920 0.77 KIT (0.45) KITACACB
SCHEMBL14754780 0.77 KIT (0.45) KITACACB
SCHEMBL12550473 0.77 ACACB (0.53) ACACB
SCHEMBL12572042 0.77 POLB (0.53) KITACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011067306-A1 CYCLOHEXANE DERIVATIVES AS INHIBITORS OF ACETYL-COA CARBOXYLASE (ACC) NOVARTIS AG (CH) 2011-06-09 WO disclosed