SCHEMBL12576506

SCHEMBL12576506

CC[C@H](Nc1c(Nc2cccc(C(=O)N(C)C)c2O)c(=O)c1=O)c1ccc(C)cc1

nearest known ligand 0.85

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 20/20 0.85
CXCR1 P25024 12/20 0.85
CCR7 P32248 1/20 0.72
CCR6 P51684 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12576508 1.00 CXCR2 (0.85) CXCR2CXCR1CCR7CCR6
SCHEMBL14511214 0.93 CXCR2 (0.86) CXCR2CXCR1
SCHEMBL12262251 0.92 CXCR2 (1.00) CXCR2CXCR1
SCHEMBL247103 0.92 CXCR2 (1.00) CXCR2CXCR1
SCHEMBL12262217 0.92 CXCR2 (1.00) CXCR2CXCR1
SCHEMBL12262254 0.91 CXCR2 (0.83) CXCR2CXCR1
SCHEMBL12086692 0.91 CXCR2 (0.88) CXCR2CXCR1CCR7CCR6
SCHEMBL12262259 0.91 CXCR2 (0.84) CXCR2CXCR1
SCHEMBL12086827 0.91 CXCR2 (0.84) CXCR2CXCR1
SCHEMBL12576503 0.90 CXCR2 (0.81) CXCR2CXCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7964646-B2 3,4-DI-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands SCHERING CORPORATION (US) 2011-06-21 US disclosed