SCHEMBL12576509

SCHEMBL12576509

Cc1ccc([C@H](C)Nc2c(Nc3cccc(C(=O)N(C)C)c3O)c(=O)c2=O)cc1

nearest known ligand 0.84

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 18/20 0.84
CXCR1 P25024 10/20 0.84
CCR6 P51684 2/20 0.66
CCR7 P32248 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12576507 1.00 CXCR2 (0.84) CXCR2CXCR1CCR6CCR7
SCHEMBL248295 0.91 CXCR2 (1.00) CXCR2CXCR1CCR6CCR7
SCHEMBL12262239 0.91 CXCR2 (1.00) CXCR2CXCR1CCR6CCR7
SCHEMBL12086787 0.91 CXCR2 (1.00) CXCR2CXCR1CCR6CCR7
SCHEMBL12262243 0.90 CXCR2 (0.82) CXCR2CXCR1CCR6
SCHEMBL12262246 0.90 CXCR2 (0.82) CXCR2CXCR1CCR6
SCHEMBL13591138 0.89 CXCR2 (0.79) CXCR2CXCR1CCR6
SCHEMBL12262102 0.88 CXCR2 (0.66) CXCR2CXCR1CCR6CCR7
SCHEMBL12262224 0.88 CXCR2 (0.82) CXCR2CXCR1CCR6CCR7
SCHEMBL12576506 0.86 CXCR2 (0.85) CXCR2CXCR1CCR6CCR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7964646-B2 3,4-DI-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands SCHERING CORPORATION (US) 2011-06-21 US disclosed