SCHEMBL12595293

SCHEMBL12595293

CC1NC(=O)c2cc3ccc(C(=O)Nc4nc5ccccc5n4CCCN(C)C)nc3n2C1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RPS6KA3 P51812 13/20 1.00
RPS6KA2 Q15349 9/20 0.78
PRKD3 O94806 1/20 0.60
ADRB2 P07550 1/20 0.60
RET P07949 1/20 0.60
PDGFRA P16234 1/20 0.60
FGFR2 P21802 1/20 0.60
ADORA2A P29274 1/20 0.60
ADRA1A P35348 1/20 0.60
ADRA1B P35368 1/20 0.60
FLT3 P36888 1/20 0.60
CLK1 P49759 1/20 0.60
CLK2 P49760 1/20 0.60
PRKD1 Q15139 1/20 0.60
LRRK2 Q5S007 1/20 0.60
PRKD2 Q9BZL6 1/20 0.60
NISCH Q9Y2I1 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14973161 1.00 RPS6KA3 (1.00) RPS6KA3RPS6KA2PRKD3ADRB2RET
SCHEMBL14972925 1.00 RPS6KA3 (1.00) RPS6KA3RPS6KA2PRKD3ADRB2RET
SCHEMBL14972924 1.00 RPS6KA3 (1.00) RPS6KA3RPS6KA2PRKD3ADRB2RET
SCHEMBL14973160 1.00 RPS6KA3 (1.00) RPS6KA3RPS6KA2PRKD3ADRB2RET
SCHEMBL17772104 0.92 RPS6KA3 (0.86) RPS6KA3RPS6KA2PRKD3ADRB2RET
SCHEMBL14973127 0.89 RPS6KA3 (1.00) RPS6KA3RPS6KA2PRKD3ADRB2RET
SCHEMBL12595454 0.89 RPS6KA3 (1.00) RPS6KA3RPS6KA2PRKD3ADRB2RET
SCHEMBL17772103 0.89 RPS6KA3 (0.80) RPS6KA3RPS6KA2PRKD3ADRB2RET
SCHEMBL14972988 0.88 RPS6KA3 (1.00) RPS6KA3RPS6KA2
SCHEMBL1981999 0.88 RPS6KA3 (1.00) RPS6KA3RPS6KA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011071725-A1 HETEROCYCLIC COMPOUNDS CONTAINING A PYRROLOPYRIDINE OR BENZIMIDAZOLE CORE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-06-16 WO disclosed