SCHEMBL12605437

SCHEMBL12605437

CCS(=O)(=O)Nc1ccnc2[nH]ccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNNI3K Q59H18 1/20 0.48
IKBKB O14920 4/20 0.48
CHUK O15111 3/20 0.48
PTK2 Q05397 1/20 0.47
NUDT1 P36639 1/20 0.47
ROCK1 Q13464 2/20 0.46
PRKCI P41743 2/20 0.45
AXL P30530 1/20 0.45
JAK1 P23458 3/20 0.44
JAK2 O60674 1/20 0.44
TYK2 P29597 1/20 0.44
ROCK2 O75116 3/20 0.43
CIT O14578 1/20 0.43
PRKD3 O94806 1/20 0.43
MAP4K4 O95819 1/20 0.43
PRKCB P05771 1/20 0.43
PRKCA P17252 1/20 0.43
PRKACA P17612 1/20 0.43
CSNK2A2 P19784 1/20 0.43
MARK3 P27448 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30009857 0.80 JAK1 (0.57) IKBKBCHUKPTK2NUDT1ROCK1
SCHEMBL30009803 0.78 IKBKB (0.55) IKBKBCHUKROCK1PRKCIJAK1
SCHEMBL30009511 0.78 CIT (0.59) IKBKBCHUKROCK1PRKCIJAK1
SCHEMBL30009181 0.78 CIT (0.50) IKBKBCHUKNUDT1ROCK1JAK1
SCHEMBL3093132 0.78 PRKCI (0.55) TNNI3KIKBKBCHUKPTK2NUDT1
SCHEMBL30009525 0.77 IKBKB (0.76) IKBKBCHUKPTK2ROCK1JAK2
SCHEMBL30009421 0.77 JAK1 (0.46) IKBKBCHUKNUDT1ROCK1PRKCI
SCHEMBL30009164 0.77 JAK1 (0.59) IKBKBCHUKNUDT1JAK1CIT
SCHEMBL30009844 0.77 JAK1 (0.64) IKBKBCHUKROCK1JAK1CIT
SCHEMBL30009186 0.74 JAK1 (0.60) IKBKBCHUKPTK2NUDT1ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7943616-B2 Protein kinase inhibitors; astham; psoriasis; antiinflammatory agents; inflammatory bowel disorders AVENTIS PHARMACEUTICALS INC. (US) 2011-05-17 US disclosed