SCHEMBL12629652

SCHEMBL12629652

O=C(O)c1cnc(-c2ccc3c(Nc4ncc(C(F)(F)F)cn4)ccnc3n2)c(C(F)(F)F)c1

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 20/20 0.68
MAPK3 P27361 1/20 0.53
MAOA P21397 1/20 0.51
KCNH2 Q12809 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1858238 0.90 TRPV1 (0.65) TRPV1MAPK3MAOAKCNH2
SCHEMBL1860303 0.89 TRPV1 (0.77) TRPV1MAPK3MAOAKCNH2
SCHEMBL1863203 0.89 TRPV1 (0.66) TRPV1MAPK3MAOAKCNH2
SCHEMBL1865933 0.87 TRPV1 (0.80) TRPV1MAPK3MAOAKCNH2
SCHEMBL1858241 0.85 TRPV1 (0.58) TRPV1MAPK3MAOAKCNH2
SCHEMBL1859378 0.84 TRPV1 (0.73) TRPV1MAPK3MAOAKCNH2
SCHEMBL1856817 0.84 TRPV1 (0.69) TRPV1MAPK3MAOAKCNH2
SCHEMBL12629706 0.82 TRPV1 (0.69) TRPV1MAPK3MAOAKCNH2
SCHEMBL1860616 0.82 TRPV1 (0.69) TRPV1MAPK3MAOAKCNH2
SCHEMBL1866427 0.82 TRPV1 (0.54) TRPV1MAOAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7935702-B2 Substituted biaryl quinolin-4-ylamine analogues NEUROGEN CORPORATION (US) 2011-05-03 US disclosed
US-7935702-B2 Substituted biaryl quinolin-4-ylamine analogues NEUROGEN CORPORATION (US) 2011-05-03 US disclosed