SCHEMBL12656264

SCHEMBL12656264

C=CCn1c(=O)oc2cc3c(O)c(c21)C[C@@H](C)CC[C@H](O)[C@@H](C)/C=C(\C)[C@H](OC(N)=O)[C@@H](OC)/C=C\C=C(/C)C(=O)N3

nearest known ligand 0.85

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 17/20 0.85
HSP90AB1 P08238 8/20 0.85
PDGFRA P16234 1/20 0.58
ALDH1A1 P00352 1/20 0.43
ERBB2 P04626 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12017386 1.00 HSP90AA1 (0.85) HSP90AA1HSP90AB1PDGFRAALDH1A1ERBB2
SCHEMBL13215948 0.92 HSP90AA1 (1.00) HSP90AA1HSP90AB1PDGFRAALDH1A1ERBB2
SCHEMBL13037483 0.92 HSP90AA1 (1.00) HSP90AA1HSP90AB1PDGFRAALDH1A1ERBB2
SCHEMBL255010 0.92 HSP90AA1 (1.00) HSP90AA1HSP90AB1PDGFRAALDH1A1ERBB2
SCHEMBL140262 0.88 HSP90AA1 (0.92) HSP90AA1HSP90AB1PDGFRAALDH1A1ERBB2
SCHEMBL13037450 0.87 HSP90AA1 (0.90) HSP90AA1HSP90AB1PDGFRAALDH1A1ERBB2
SCHEMBL15160217 0.85 HSP90AA1 (0.87) HSP90AA1HSP90AB1PDGFRAALDH1A1ERBB2
SCHEMBL12656260 0.83 HSP90AA1 (0.87) HSP90AA1HSP90AB1PDGFRAALDH1A1ERBB2
SCHEMBL14370485 0.83 HSP90AA1 (0.83) HSP90AA1HSP90AB1PDGFRAALDH1A1ERBB2
SCHEMBL140125 0.82 HSP90AA1 (0.82) HSP90AA1HSP90AB1PDGFRAALDH1A1ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716119-B1 Analogs of benzoquinone-containing ansamycins for the treatment of cancer INFINITY DISCOVERY INC (US) 2013-03-06 EP disclosed
WO-2011060328-A1 COMPOSITIONS, KITS, AND METHODS FOR IDENTIFICATION, ASSESSMENT, PREVENTION, AND THERAPY OF CANCER INFINITY PHARMACEUTICALS, INC. (US) 2011-05-19 WO disclosed
WO-2010135426-A1 METHODS OF TREATING LIPOSARCOMA INFINITY PHARMACEUTICALS, INC. (US) 2010-11-25 WO disclosed
EP-1904057-B1 HYDROQUINONE ANSAMYCINS IN THE TREATMENT OF GASTROINTESTINAL STROMAL TUMORS INFINITY DISCOVERY INC (US) 2009-12-16 EP disclosed