SCHEMBL12677271

SCHEMBL12677271

CNC(=O)CNc1nc2oc(-c3ccc(C4(N(C)Cl)CCC4)cc3)c(-c3ccccc3)c2c(=O)n1C

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TNK2 Q07912 9/20 0.36
CHEK1 O14757 1/20 0.35
OPRM1 P35372 8/20 0.34
OPRL1 P41146 6/20 0.34
LCK P06239 3/20 0.33
AURKA O14965 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14235797 0.88 TNK2 (0.38) TNK2CHEK1OPRM1OPRL1LCK
SCHEMBL12095402 0.87 AKT1 (0.41) TNK2CHEK1
Hydrochloric Acid SCHEMBL1900324 0.87 AKT1 (0.40) TNK2CHEK1
SCHEMBL1903880 0.86 TNK2 (0.37) TNK2CHEK1OPRM1OPRL1LCK
SCHEMBL14119016 0.82 AKT1 (0.40) TNK2CHEK1LCKAURKA
SCHEMBL1906685 0.79 AKT1 (0.39) CHEK1
SCHEMBL1904617 0.77 CHEK1 (0.36) TNK2CHEK1OPRM1LCKAURKA
SCHEMBL1904185 0.76 AURKA (0.37) TNK2CHEK1LCKAURKA
SCHEMBL1904665 0.75 AKT1 (0.40)
SCHEMBL1901112 0.75 CHEK1 (0.43) CHEK1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011055115-A1 AKT / PKB INHIBITORS ALMAC DISCOVERY LIMITED (GB) 2011-05-12 WO disclosed