SCHEMBL12694308

SCHEMBL12694308

COc1cc2ncnc(Nc3ccc(NC(=O)NCCCCN4CCCC4)cc3)c2cc1OCCCN1CCOCC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 14/20 0.72
KDR P35968 13/20 0.72
SRC P12931 3/20 0.72
AURKA O14965 2/20 0.72
AURKB Q96GD4 2/20 0.72
ROCK2 O75116 1/20 0.72
ALDH1A1 P00352 1/20 0.72
LCK P06239 1/20 0.72
FYN P06241 1/20 0.72
RET P07949 1/20 0.72
MET P08581 1/20 0.72
MAPT P10636 1/20 0.72
PDGFRA P16234 1/20 0.72
LTK P29376 1/20 0.72
TTK P33981 1/20 0.72
MAP2K2 P36507 1/20 0.72
MAP2K1 Q02750 1/20 0.72
BTK Q06187 1/20 0.72
TYRO3 Q06418 1/20 0.72
TNK2 Q07912 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12694382 0.94 EGFR (0.79) EGFRKDRSRCAURKAAURKB
SCHEMBL12694354 0.90 KDR (0.64) EGFRKDRSRCAURKAAURKB
SCHEMBL12694381 0.89 EGFR (0.73) EGFRKDRSRCAURKAAURKB
SCHEMBL25739558 0.87 EGFR (0.72) EGFRKDRSRCAURKAAURKB
SCHEMBL12694349 0.86 AURKA (0.76) EGFRKDRSRCAURKAAURKB
SCHEMBL12694312 0.86 EGFR (0.79) EGFRKDRSRCAURKAAURKB
SCHEMBL12694306 0.86 AURKA (0.76) EGFRKDRSRCAURKAAURKB
SCHEMBL12694307 0.85 EGFR (0.93) EGFRKDRSRCAURKAAURKB
SCHEMBL12694385 0.84 EGFR (0.73) EGFRKDRSRCAURKAAURKB
SCHEMBL6704281 0.84 EGFR (0.80) EGFRKDRSRCAURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012089137-A1 ARYLUREA COMPOUND, INTERMEDIATE AND USE THEREOF 上海医药工业研究院 (CN) 2012-07-05 WO disclosed