SCHEMBL12694370

SCHEMBL12694370

COc1cc2ncnc(Nc3cccc(NC(=O)Nc4cccc(F)c4)c3)c2cc1OCCCN1CCOCC1

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.85
KDR P35968 11/20 0.85
BRAF P15056 5/20 0.85
AURKA O14965 3/20 0.74
SRC P12931 3/20 0.72
HDAC1 Q13547 3/20 0.68
HDAC3 O15379 2/20 0.68
HDAC6 Q9UBN7 2/20 0.68
LCK P06239 2/20 0.68
RET P07949 2/20 0.68
MET P08581 2/20 0.68
MAPT P10636 2/20 0.68
LTK P29376 2/20 0.68
TNK2 Q07912 2/20 0.68
MAP4K5 Q9Y4K4 2/20 0.68
ROCK2 O75116 1/20 0.68
ALDH1A1 P00352 1/20 0.68
FYN P06241 1/20 0.68
PDGFRA P16234 1/20 0.68
TTK P33981 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12694392 0.92 EGFR (1.00) EGFRKDRBRAFAURKASRC
SCHEMBL12694406 0.91 BRAF (1.00) EGFRKDRBRAFAURKASRC
SCHEMBL12694377 0.89 EGFR (0.81) EGFRKDRBRAFAURKASRC
SCHEMBL12694363 0.88 EGFR (0.80) EGFRKDRBRAFAURKASRC
SCHEMBL12694307 0.88 EGFR (0.93) EGFRKDRBRAFAURKASRC
SCHEMBL2049532 0.88 PDGFRB (0.78) EGFRKDRBRAFAURKASRC
SCHEMBL12694382 0.88 EGFR (0.79) EGFRKDRBRAFAURKASRC
SCHEMBL12694386 0.88 EGFR (1.00) EGFRKDRBRAFAURKASRC
SCHEMBL12694376 0.87 EGFR (0.78) EGFRKDRBRAFAURKASRC
SCHEMBL31167326 0.87 EGFR (0.78) EGFRKDRBRAFAURKASRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012089137-A1 ARYLUREA COMPOUND, INTERMEDIATE AND USE THEREOF 上海医药工业研究院 (CN) 2012-07-05 WO disclosed