SCHEMBL12700481

SCHEMBL12700481

Cc1cc(C)nc(N2CCC3(CC2)NCCN(Cc2nn(C)cc2-c2ccc(N)cc2)C3=O)n1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 12/20 0.61
HCRTR2 O43614 12/20 0.61
CDK8 P49336 3/20 0.32
CDK19 Q9BWU1 3/20 0.32
CCNC P24863 2/20 0.32
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30
SCN9A Q15858 2/20 0.30
HAVCR2 Q8TDQ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9948786 0.91 HCRTR1 (0.72) HCRTR1HCRTR2KDM4EALDH1A1HPGD
SCHEMBL9949217 0.90 HCRTR1 (0.59) HCRTR1HCRTR2HPGDHSD17B10
SCHEMBL9949033 0.90 HCRTR1 (0.59) HCRTR1HCRTR2
SCHEMBL9948904 0.89 HCRTR1 (0.57) HCRTR1HCRTR2CDK8CDK19CCNC
SCHEMBL9949343 0.87 HCRTR1 (0.62) HCRTR1HCRTR2KDM4E
SCHEMBL9948825 0.87 HCRTR1 (0.55) HCRTR1HCRTR2KDM4EALDH1A1HPGD
SCHEMBL9949052 0.86 HCRTR1 (0.55) HCRTR1HCRTR2KDM4E
SCHEMBL9948796 0.86 HCRTR1 (0.59) HCRTR1HCRTR2KDM4EALDH1A1HPGD
SCHEMBL9948746 0.86 HCRTR2 (0.60) HCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL9948768 0.86 HCRTR2 (0.60) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012101487-A1 DI/TRI-AZA-SPIRO-C9-C11ALKANES NOVARTIS AG (CH) 2012-08-02 WO disclosed