SCHEMBL12717138

SCHEMBL12717138

SCc1ccc(-c2c(Cl)nc(Cl)nc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.50
KDM4E B2RXH2 4/20 0.37
ALDH1A1 P00352 3/20 0.37
CYP1A2 P05177 2/20 0.37
MAPK1 P28482 2/20 0.37
HSD17B10 Q99714 2/20 0.37
MAPT P10636 2/20 0.37
LMNA P02545 4/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
HEXA P06865 2/20 0.35
HEXB P07686 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
SLC22A1 O15245 1/20 0.35
DHFR P00374 1/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA2A P08913 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12717320 0.89 KDM4E (0.46) IDO1KDM4EALDH1A1CYP1A2MAPT
SCHEMBL4841423 0.87 KDM4E (0.46) KDM4EALDH1A1CYP1A2MAPK1HSD17B10
SCHEMBL1572963 0.80 KDM4E (0.55) KDM4EALDH1A1CYP1A2MAPK1HSD17B10
SCHEMBL1572910 0.80 KDM4E (0.55) KDM4EALDH1A1CYP1A2MAPK1HSD17B10
SCHEMBL1573080 0.79 KDM4E (0.49) KDM4EALDH1A1CYP1A2MAPK1HSD17B10
SCHEMBL11864905 0.75 CYP1A2 (0.57) KDM4EALDH1A1CYP1A2MAPK1HSD17B10
SCHEMBL1573037 0.75 MAPT (0.41) KDM4EALDH1A1CYP1A2MAPK1HSD17B10
SCHEMBL1573115 0.72 KDM4E (0.61) KDM4EALDH1A1MAPTLMNAMEN1
SCHEMBL14313984 0.72 KDM4E (0.44) IDO1KDM4EALDH1A1MAPTLMNA
SCHEMBL307618 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542978-B1 NOVEL BIO-ACTIVE MOLECULES ORCHID RES LAB LTD (IN) 2011-04-13 EP disclosed
US-7317014-B2 Bio-active pyrimidine molecules ORCHID RESEARCH LABORATORIES, LTD. (IN) 2008-01-08 US disclosed