SCHEMBL127220

SCHEMBL127220

C/C(=C\c1c(Cl)cc(Cl)cc1Cl)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.44
APEX1 P27695 3/20 0.40
AKR1C4 P17516 1/20 0.38
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38
TPMT P51580 1/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
MAPK1 P28482 1/20 0.35
BLM P54132 1/20 0.35
PMP22 Q01453 1/20 0.35
KMT2A Q03164 1/20 0.35
TSHR P16473 2/20 0.35
CASP1 P29466 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
RECQL P46063 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL127221 1.00 AKR1C3 (0.44) AKR1C3APEX1AKR1C4AKR1C2AKR1C1
SCHEMBL3069068 0.86 AKR1C3 (0.42) AKR1C3APEX1LMNAALDH1A1
SCHEMBL3069073 0.86 AKR1C3 (0.42) AKR1C3APEX1LMNAALDH1A1
SCHEMBL19967035 0.86 AKR1C3 (0.42) AKR1C3APEX1TPMTMEN1LMNA
SCHEMBL16224162 0.85 TTR (0.48) AKR1C3APEX1TPMTTSHR
SCHEMBL15199397 0.85 TTR (0.48) AKR1C3APEX1TPMTTSHR
SCHEMBL21470298 0.82 EIF4A3 (0.42) AKR1C3APEX1MAPK1
SCHEMBL7820417 0.80 AKR1C3 (0.53) AKR1C3APEX1MEN1LMNACYP1A2
SCHEMBL7820420 0.80 AKR1C3 (0.53) AKR1C3APEX1MEN1LMNACYP1A2
SCHEMBL10744557 0.78 AKR1C3 (0.55) AKR1C3APEX1TPMTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 61 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0841380-B1 Method of making polymeric binders and use thereof in antifouling paints WITCO GMBH (DE) 1999-08-25 EP claimed
EP-0841380-A1 Method of making polymeric binders and use thereof in antifouling paints Witco GmbH (DE) 1998-05-13 EP claimed
EP-2531889-B1 USE OF A PHOTOPOLYMER FORMULATION WITH ESTER-BASED WRITING MONOMERS FOR THE FABRICATION OF HOLOGRAPHIC MEDIA COVESTRO DEUTSCHLAND AG (DE) 2020-06-03 EP disclosed
EP-2638544-B1 PHOTOPOLYMER FORMULATION FOR PRODUCING HOLOGRAPHIC MEDIA HAVING HIGHLY CROSS-LINKED MATRIX POLYMERS COVESTRO DEUTSCHLAND AG (DE) 2018-12-26 EP disclosed
EP-2904531-B1 METHOD FOR SELECTING PHOTOINITIATOR SYSTEMS COVESTRO DEUTSCHLAND AG (DE) 2018-12-19 EP disclosed
EP-2342249-B1 PREPOLYMER-BASED POLYURETHANE FORMULATIONS FOR PRODUCING HOLOGRAPHIC MEDIA COVESTRO DEUTSCHLAND AG (DE) 2017-10-25 EP disclosed
EP-2342254-B1 MEDIA FOR VOLUME-HOLOGRAPHIC RECORDING BASED ON SELF-DEVELOPING POLYMERS COVESTRO DEUTSCHLAND AG (DE) 2017-09-27 EP disclosed
EP-2962302-B1 PROTECTIVE VARNISHES FOR PHOTOPOLYMER APPLICATIONS AN ACRYLATE BASIS COVESTRO DEUTSCHLAND AG (DE) 2017-06-14 EP disclosed
EP-2888116-B1 SECURITY AND/OR VALUE DOCUMENT CONTAINING A VISUAL SWITCHABLE WINDOW WITH A HOLOGRAM COVESTRO DEUTSCHLAND AG (DE) 2016-09-21 EP disclosed
EP-2845195-B1 NEW PHOTOINITIATORS FOR PHOTOPOLYMERS COVESTRO DEUTSCHLAND AG (DE) 2016-07-13 EP disclosed
EP-2172502-B1 POLYETHER-BASED POLYURETHANE FORMULATIONS FOR PRODUCING HOLOGRAPHIC MEDIA COVESTRO DEUTSCHLAND AG (DE) 2016-04-20 EP disclosed
WO-2010037496-A1 PREPOLYMER-BASED POLYURETHANE FORMULATIONS FOR PRODUCING HOLOGRAPHIC MEDIA BAYER MATERIALSCIENCE AG (DE) 2010-04-08 WO disclosed
EP-2172504-A1 Photopolymer formulations with low interlacing density Bayer MaterialScience AG (DE) 2010-04-07 EP disclosed
EP-2172503-A1 Special polyether-based polyurethane formulations for producing holographic media Bayer MaterialScience AG (DE) 2010-04-07 EP disclosed
EP-2172502-A1 Polyether-based polyurethane formulations for producing holographic media Bayer MaterialScience AG (DE) 2010-04-07 EP disclosed
US-6432498-B1 Volume hologram laminate DAI NIPPON PRINTING CO., LTD. (JP) 2002-08-13 US disclosed
EP-0841380-B1 Method of making polymeric binders and use thereof in antifouling paints WITCO GMBH (DE) 1999-08-25 EP disclosed
EP-0841380-A1 Method of making polymeric binders and use thereof in antifouling paints Witco GmbH (DE) 1998-05-13 EP disclosed
EP-0833870-A1 POLYMERS FOR ANTIFOULING COATINGS AND A PROCESS FOR THE PREPARATION THEREOF Jotun A/S (NO) 1998-04-08 EP disclosed
WO-1996041842-A1 POLYMERS FOR ANTIFOULING COATINGS AND A PROCESS FOR THE PREPARATION THEREOF JOTUN A/S (NO) 1996-12-27 WO disclosed