SCHEMBL12724898

SCHEMBL12724898

COc1cc(O)cc(Nc2ncc3ccc(OC4CCN(C(C)C)CC4)cc3n2)c1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 16/20 0.43
CDK4 P11802 1/20 0.41
CCND1 P24385 1/20 0.41
CDK6 Q00534 1/20 0.41
CCNA2 P20248 2/20 0.39
CDK2 P24941 2/20 0.39
CDK7 P50613 2/20 0.39
CCNH P51946 2/20 0.39
MNAT1 P51948 2/20 0.39
CHEK1 O14757 1/20 0.39
CCNK O75909 1/20 0.38
CDK12 Q9NYV4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1634242 0.94 HRH3 (0.44) HRH3CDK4CCND1CDK6CCNA2
SCHEMBL12724903 0.90 CDK4 (0.47) CDK4CCND1CDK6CCNA2CDK2
SCHEMBL12724921 0.87 SYK (0.44) HRH3CDK4CCND1CDK6
SCHEMBL1632964 0.87 USP2 (0.49) CCNA2CDK2
SCHEMBL13498327 0.85 IKBKB (0.43) CHEK1
SCHEMBL1633930 0.84 HRH3 (0.43) HRH3CDK4CCND1CDK6
SCHEMBL1632568 0.84 HRH3 (0.43) HRH3CDK4CCND1CDK6
SCHEMBL1634267 0.83 CDK4 (0.50) CDK4CCND1CDK6CCNA2CDK2
SCHEMBL1633595 0.82 HRH3 (0.43) HRH3CDK4CCND1CDK6
SCHEMBL1634281 0.81 HRH3 (0.48) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7932262-B2 Quinazolines for PDK1 inhibition NOVARTIS AG (CH) 2011-04-26 US disclosed