SCHEMBL12799990

SCHEMBL12799990

C[S+]([O-])c1cc(C2(NC(=O)c3cncc4c3cnn4-c3ccc(F)cc3)CC2)ccn1

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 20/20 0.73
KCNH2 Q12809 2/20 0.73
ADRB1 P08588 1/20 0.73
CYP3A4 P08684 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670683 0.85 CCR1 (0.76) CCR1KCNH2ADRB1CYP3A4
Bi 639667 SCHEMBL1670702 0.84 CCR1 (1.00) CCR1KCNH2ADRB1CYP3A4
SCHEMBL1670357 0.84 CCR1 (0.73) CCR1KCNH2ADRB1CYP3A4
SCHEMBL1670833 0.83 CCR1 (0.71) CCR1KCNH2ADRB1CYP3A4
SCHEMBL1670643 0.82 CCR1 (0.77) CCR1KCNH2ADRB1CYP3A4
SCHEMBL13556701 0.82 CCR1 (0.76) CCR1KCNH2ADRB1CYP3A4
SCHEMBL1670697 0.82 CCR1 (0.70) CCR1KCNH2ADRB1CYP3A4
SCHEMBL1670930 0.81 CCR1 (1.00) CCR1KCNH2ADRB1CYP3A4
SCHEMBL1671964 0.81 CCR1 (0.69) CCR1KCNH2ADRB1CYP3A4
SCHEMBL1672930 0.81 CCR1 (0.68) CCR1KCNH2ADRB1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011049917-A1 INDAZOLE AND PYRAZOLOPYRIDINE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-04-28 WO disclosed