SCHEMBL12801098

SCHEMBL12801098

CC(=O)Nc1ccc(-c2ccnc(Nc3ccc(N4CCOCC4)cc3)n2)cc1N

nearest known ligand 0.76

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 20/20 0.76
JAK3 P52333 10/20 0.65
JAK1 P23458 4/20 0.62
TYK2 P29597 4/20 0.61
HDAC3 O15379 1/20 0.61
NCOR1 O75376 1/20 0.61
HDAC1 Q13547 1/20 0.61
HDAC2 Q92769 1/20 0.61
HDAC8 Q9BY41 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12800935 0.90 JAK2 (0.69) JAK2JAK3JAK1TYK2HDAC3
SCHEMBL12522201 0.90 JAK2 (0.63) JAK2JAK3JAK1TYK2HDAC3
SCHEMBL12801620 0.89 JAK2 (0.66) JAK2JAK3JAK1TYK2HDAC3
SCHEMBL12801381 0.89 JAK2 (0.62) JAK2JAK3JAK1TYK2HDAC3
SCHEMBL12522331 0.88 JAK2 (0.64) JAK2JAK3JAK1TYK2HDAC3
SCHEMBL12801263 0.88 JAK2 (0.71) JAK2JAK3JAK1TYK2HDAC3
SCHEMBL12522359 0.88 JAK2 (0.61) JAK2JAK3JAK1TYK2HDAC3
SCHEMBL12801354 0.87 JAK2 (0.65) JAK2JAK3JAK1TYK2HDAC3
SCHEMBL12801350 0.87 JAK2 (0.65) JAK2JAK3JAK1TYK2HDAC3
SCHEMBL12274521 0.87 JAK2 (0.72) JAK2JAK3JAK1TYK2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed