SCHEMBL12809013

SCHEMBL12809013

CC(C)Oc1ccc(-c2nc(-c3cccc4nn(CCC=O)cc34)no2)cc1Cl

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.56
CYP2C9 P11712 1/20 0.54
S1PR3 Q99500 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12601257 0.94 S1PR1 (0.54) S1PR1CYP2C9S1PR3
SCHEMBL1398466 0.88 S1PR1 (0.71) S1PR1CYP2C9S1PR3
SCHEMBL1398430 0.87 S1PR1 (0.68) S1PR1CYP2C9S1PR3
SCHEMBL2048791 0.86 S1PR1 (0.67) S1PR1CYP2C9S1PR3
SCHEMBL2054001 0.85 S1PR1 (0.59) S1PR1CYP2C9S1PR3
SCHEMBL1398629 0.85 S1PR1 (0.59) S1PR1CYP2C9S1PR3
SCHEMBL13644176 0.85 S1PR1 (0.54) S1PR1S1PR3
SCHEMBL1981338 0.84 S1PR1 (0.58) S1PR1CYP2C9S1PR3
SCHEMBL1398517 0.84 S1PR1 (0.57) S1PR1CYP2C9S1PR3
SCHEMBL2054003 0.78 S1PR1 (0.64) S1PR1CYP2C9S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137181-B1 OXADIAZOLE SUBSTITUTED INDAZOLE DERIVATIVES FOR USE AS SPHINGOSINE 1-PHOSPHATE (S1P) AGONISTS GLAXO GROUP LTD (GB) 2011-03-02 EP disclosed