SCHEMBL12812352

SCHEMBL12812352

NO[C@@H]1CC[C@@H](c2cccc(F)c2F)CN(C(=O)NC2CC2)C1

nearest known ligand 0.46

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 14/20 0.46
HCRTR2 O43614 5/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12812353 0.97 CALCRL (0.45) CALCRLHCRTR2
SCHEMBL12812342 0.86 HCRTR2 (0.42) CALCRLHCRTR2
SCHEMBL12812347 0.85 HCRTR2 (0.41) CALCRLHCRTR2
SCHEMBL12812345 0.84 HCRTR2 (0.42) CALCRLHCRTR2
SCHEMBL12812350 0.82 HCRTR2 (0.43) CALCRLHCRTR2
SCHEMBL12812343 0.81 NAMPT (0.41) CALCRLHCRTR2
SCHEMBL12812348 0.80 HCRTR2 (0.41) CALCRLHCRTR2
SCHEMBL12812368 0.78 HCRTR2 (0.41) CALCRLHCRTR2
SCHEMBL12812340 0.75 HCRTR2 (0.39) CALCRLHCRTR2
SCHEMBL12812351 0.74 HCRTR2 (0.42) CALCRLHCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1804919-B1 CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2011-03-30 EP disclosed