SCHEMBL12812481

SCHEMBL12812481

Cc1cc(-c2ccc3ncc(N4CCN(Cc5cccc(N)c5)CC4)nc3c2)cc(C)c1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44
MELK Q14680 1/20 0.38
MAPT P10636 1/20 0.37
HCRTR1 O43613 2/20 0.37
HCRTR2 O43614 2/20 0.37
DRD2 P14416 3/20 0.37
DRD4 P21917 3/20 0.37
DRD3 P35462 3/20 0.37
HTR1A P08908 1/20 0.37
HTR1D P28221 1/20 0.37
HTR1B P28222 1/20 0.37
RAD52 P43351 1/20 0.36
BCL2L1 Q07817 1/20 0.36
DHFR P00374 1/20 0.36
HTR3A P46098 1/20 0.36
HRH4 Q9H3N8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12812482 0.90 NPC1 (0.49) NPC1RAB9AALDH1A1KDM4EPOLB
SCHEMBL10179172 0.89 NPC1 (0.63) NPC1RAB9AALDH1A1KDM4EPOLB
SCHEMBL1441771 0.89 NPC1 (0.52) NPC1RAB9AALDH1A1KDM4EPOLB
SCHEMBL12812430 0.89 NPC1 (0.53) NPC1RAB9AALDH1A1KDM4EPOLB
SCHEMBL1442613 0.86 NPC1 (0.47) NPC1RAB9AALDH1A1KDM4EPOLB
SCHEMBL1443431 0.86 NPC1 (0.58) NPC1RAB9AALDH1A1KDM4EPOLB
SCHEMBL10178977 0.86 NPC1 (0.50) NPC1RAB9AALDH1A1KDM4EPOLB
SCHEMBL1442823 0.84 NPC1 (0.49) NPC1RAB9AALDH1A1KDM4EPOLB
SCHEMBL1442658 0.83 MAPT (0.43) NPC1RAB9AALDH1A1KDM4EPOLB
SCHEMBL1442719 0.82 NPC1 (0.49) NPC1RAB9AALDH1A1KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011026579-A1 SUBSTITUTED AMINOQUINOXALINES AS TYROSINE THREONINE KINASE INHIBITORS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-03-10 WO disclosed