SCHEMBL12820035

SCHEMBL12820035

CN(C)CCNC(=O)O[C@H]1CC[C@H](Nc2cc(-c3c4n(c5ccccc35)C(=O)CC(C)(C)C4)ccc2C=O)CC1

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 4/20 0.32
HSP90AB1 P08238 4/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31
EGFR P00533 1/20 0.31
SRC P12931 1/20 0.31
PTGER4 P35408 1/20 0.30
MELK Q14680 1/20 0.30
ACACB O00763 1/20 0.30
ACACA Q13085 1/20 0.30
NPY1R P25929 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12820161 0.89 HSP90AA1 (0.43) HSP90AA1HSP90AB1
SCHEMBL12820409 0.85 HSP90AA1 (0.37) HSP90AA1HSP90AB1KDM4EALDH1A1HPGD
SCHEMBL12820391 0.82 HSP90AA1 (0.42) HSP90AA1HSP90AB1
SCHEMBL12820133 0.82 HSP90AA1 (0.43) HSP90AA1HSP90AB1
SCHEMBL12820487 0.81 HSP90AA1 (0.42) HSP90AA1HSP90AB1
SCHEMBL12820416 0.79 HSP90AA1 (0.37) HSP90AA1HSP90AB1
SCHEMBL12819930 0.78 HSP90AA1 (0.44) HSP90AA1HSP90AB1
SCHEMBL12819524 0.78 HSP90AA1 (0.42) HSP90AA1HSP90AB1
SCHEMBL12820144 0.78 HSP90AA1 (0.47) HSP90AA1HSP90AB1
SCHEMBL12819856 0.77 HSP90AA1 (0.43) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011035417-A1 HSP-90 BINDING COMPOUNDS, COMPOSITIONS THEREOF, AND THEIR USE FN THE TREATMENT OF AUTOIMMUNE AND INFLAMMATORY DISEASES AEGERA THERAPEUTICS INC. (CA) 2011-03-31 WO disclosed