SCHEMBL12835643

SCHEMBL12835643

Cc1nnc(C2C3CN(C(=O)OC(C)(C)C)C[C@@H]32)o1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.48
GPR119 Q8TDV5 1/20 0.42
NR1H2 P55055 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.38
GAA P10253 1/20 0.38
THRB P10828 1/20 0.38
USP2 O75604 1/20 0.38
SSTR4 P31391 1/20 0.38
ALDH1A1 P00352 1/20 0.37
JAK3 P52333 1/20 0.37
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
NAMPT P43490 1/20 0.37
MAPT P10636 2/20 0.36
HSD11B1 P28845 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9965957 1.00 KDM5A (0.48) KDM5AGPR119NR1H2SMN1; SMN2GAA
SCHEMBL16182224 1.00 KDM5A (0.48) KDM5AGPR119NR1H2SMN1; SMN2GAA
SCHEMBL14641877 0.86 NR1H2 (0.40) KDM5ANR1H2SMN1; SMN2GAATHRB
SCHEMBL9963083 0.86 NR1H2 (0.40) KDM5ANR1H2SMN1; SMN2GAATHRB
SCHEMBL24824540 0.86 SMN1; SMN2 (0.44) GPR119NR1H2SMN1; SMN2GAATHRB
SCHEMBL9965918 0.85 SMN1; SMN2 (0.47) GPR119NR1H2SMN1; SMN2GAATHRB
SCHEMBL12835905 0.83 NR1H2 (0.40) NR1H2SMN1; SMN2GAATHRBUSP2
SCHEMBL9965924 0.83 NR1H2 (0.40) NR1H2SMN1; SMN2GAATHRBUSP2
SCHEMBL9965923 0.80 NR1H2 (0.38) NR1H2SMN1; SMN2GAATHRBUSP2
SCHEMBL16182181 0.80 NR1H2 (0.38) NR1H2SMN1; SMN2GAATHRBUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011025690-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2011-03-03 WO disclosed