SCHEMBL12837784

SCHEMBL12837784

CC[C@@H]1c2nncn2-c2cnc(N[C@@H](C)c3ccc(C)cc3)nc2N1C1CCCC1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 7/20 0.60
PLK1 P53350 18/20 0.40
PLK3 Q9H4B4 12/20 0.40
PLK2 Q9NYY3 12/20 0.40
TAF1 P21675 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2360486 0.92 BRD4 (0.59) BRD4PLK1PLK3PLK2TAF1
SCHEMBL523873 0.92 BRD4 (0.59) BRD4PLK1PLK3PLK2TAF1
SCHEMBL20815326 0.92 BRD4 (0.59) BRD4PLK1PLK3PLK2TAF1
SCHEMBL523874 0.92 BRD4 (0.59) BRD4PLK1PLK3PLK2TAF1
SCHEMBL10313789 0.92 BRD4 (0.59) BRD4PLK1PLK3PLK2TAF1
SCHEMBL523203 0.92 BRD4 (0.66) BRD4PLK1PLK3PLK2
SCHEMBL524306 0.92 BRD4 (0.66) BRD4PLK1PLK3PLK2
SCHEMBL524305 0.92 BRD4 (0.66) BRD4PLK1PLK3PLK2
SCHEMBL20815288 0.88 BRD4 (0.55) BRD4PLK1PLK3PLK2TAF1
SCHEMBL524048 0.88 BRD4 (0.55) BRD4PLK1PLK3PLK2TAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011038185-A2 METHODS FOR PREPARING PYRIMIDINE DERIVATIVES USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-03-31 WO disclosed