SCHEMBL12850319

SCHEMBL12850319

NC1(COc2cncc(-c3cc(N[C@H]4CC[C@H](NCCF)CC4)ncc3Cl)n2)CCOCC1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 15/20 0.52
CCNK O75909 6/20 0.45
CDK9 P50750 6/20 0.45
CDK14 O94921 1/20 0.45
CDK1 P06493 1/20 0.45
CCNB1 P14635 1/20 0.45
CCNA2 P20248 1/20 0.45
CDK2 P24941 1/20 0.45
CDK7 P50613 1/20 0.45
CCNH P51946 1/20 0.45
MNAT1 P51948 1/20 0.45
CDK5 Q00535 1/20 0.45
CDK16 Q00536 1/20 0.45
CDK5R1 Q15078 1/20 0.45
CCNY Q8ND76 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12850332 0.91 CCNT1 (0.48) CCNT1CCNKCDK9CDK14CDK1
SCHEMBL15378039 0.88 CCNT1 (0.55) CCNT1CCNKCDK9CDK14CDK1
SCHEMBL15378038 0.88 CCNT1 (0.55) CCNT1CCNKCDK9CDK14CDK1
SCHEMBL8784970 0.86 CCNT1 (0.48) CCNT1CCNKCDK9CDK14CDK1
SCHEMBL12850674 0.86 CCNT1 (0.46) CCNT1CCNKCDK9CDK14CDK1
SCHEMBL12850672 0.86 CCNT1 (0.46) CCNT1CCNKCDK9CDK14CDK1
SCHEMBL12850336 0.84 CCNT1 (0.49) CCNT1
SCHEMBL12850334 0.83 CCNT1 (0.60) CCNT1CCNKCDK9CDK14CDK1
SCHEMBL12850537 0.83 CCNT1 (0.60) CCNT1CCNKCDK9CDK14CDK1
SCHEMBL12850328 0.83 CCNT1 (0.47) CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012101062-A1 SUBSTITUTED BI-HETEROARYL COMPOUNDS AS CDK9 INHIBITORS AND THEIR USES NOVARTIS AG (CH) 2012-08-02 WO disclosed