SCHEMBL12856367

SCHEMBL12856367

CC(C)CC(=O)c1ccc2c(c1)/C(=C/Nc1ccc(S(N)(=O)=O)cc1)C(=O)N2

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.43
CDK2 P24941 1/20 0.43
CA12 O43570 11/20 0.42
CA1 P00915 11/20 0.42
CA2 P00918 11/20 0.42
CA9 Q16790 11/20 0.42
KDR P35968 3/20 0.40
PDGFRB P09619 2/20 0.40
FGFR1 P11362 2/20 0.40
EGFR P00533 1/20 0.40
PDPK1 O15530 1/20 0.39
RAF1 P04049 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gw416981X SCHEMBL14040791 0.88 CDK1 (0.45) CDK1CDK2CA12CA1CA2
Gw416981X SCHEMBL5425650 0.88 CDK1 (0.45) CDK1CDK2CA12CA1CA2
Gw416981X SCHEMBL5425654 0.88 CDK1 (0.45) CDK1CDK2CA12CA1CA2
SCHEMBL7654637 0.85 TLK2 (0.47) CA12CA1CA2CA9PDPK1
SCHEMBL12856336 0.85 TLK2 (0.47) CA12CA1CA2CA9PDPK1
SCHEMBL5182747 0.84 AURKA (0.53) CA12CA1CA2CA9PDPK1
SCHEMBL12856526 0.84 AURKA (0.53) CA12CA1CA2CA9PDPK1
SCHEMBL5182752 0.84 AURKA (0.53) CA12CA1CA2CA9PDPK1
SCHEMBL12856391 0.83 AURKA (0.39) CDK1CDK2CA12CA1CA2
SCHEMBL5894173 0.83 KMT2A (0.52) CA12CA1CA2CA9KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1364212-B1 THREE HYBRID ASSAY SYSTEM GPC BIOTECH AG (DE) 2011-02-02 EP disclosed