SCHEMBL12895344

SCHEMBL12895344

Cc1ccc(C(=O)Nc2cc(C(F)(F)F)ccc2N2CCOCC2)cc1Oc1ncccc1-c1ccnc(NCCCN2CCOCC2)n1

nearest known ligand 0.81

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TEK Q02763 14/20 0.81
KDR P35968 12/20 0.81
YES1 P07947 1/20 0.54
LCK P06239 4/20 0.49
MAPK14 Q16539 3/20 0.49
JAK3 P52333 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1265603 0.90 TEK (0.80) TEKKDRYES1LCKMAPK14
SCHEMBL1264994 0.89 TEK (1.00) TEKKDRYES1LCKMAPK14
SCHEMBL2296918 0.89 TEK (0.67) TEKKDRLCKMAPK14JAK3
SCHEMBL1264439 0.83 TEK (0.88) TEKKDRYES1LCKMAPK14
SCHEMBL2297112 0.83 TEK (1.00) TEKKDR
SCHEMBL1264167 0.83 TEK (1.00) TEKKDRYES1LCKMAPK14
SCHEMBL1264886 0.83 KDR (0.70) TEKKDRYES1LCKMAPK14
SCHEMBL1264864 0.81 TEK (0.84) TEKKDRYES1LCKMAPK14
SCHEMBL1265806 0.80 TEK (0.78) TEKKDR
SCHEMBL1265761 0.78 TEK (0.76) TEKKDRYES1LCKMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7880000-B2 N-(5-(1,1- dimethylethyl)-3- isoxazolyl)-4-methyl-3- ((3-(4-pyrimidinyl)-2- pyridinyl)amino)benzamide, used for treating breast cancer or rheumatoid arthritis AMGEN INC. (US) 2011-02-01 US disclosed
US-7880000-B2 N-(5-(1,1- dimethylethyl)-3- isoxazolyl)-4-methyl-3- ((3-(4-pyrimidinyl)-2- pyridinyl)amino)benzamide, used for treating breast cancer or rheumatoid arthritis AMGEN INC. (US) 2011-02-01 US disclosed