Nicotinyl Methylamide

Nicotinyl Methylamide

SCHEMBL129458

CNC(=O)c1cccnc1

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.69
HDAC6 Q9UBN7 1/20 0.69
MKNK1 Q9BUB5 1/20 0.67
MKNK2 Q9HBH9 1/20 0.67
LMNA P02545 2/20 0.62
THRB P10828 1/20 0.62
HIF1A Q16665 1/20 0.62
ALDH1A1 P00352 4/20 0.61
ROCK2 O75116 1/20 0.61
ROCK1 Q13464 1/20 0.61
GAA P10253 3/20 0.59
APP P05067 1/20 0.59
HCAR3 P49019 1/20 0.59
HCAR2 Q8TDS4 1/20 0.59
TDP1 Q9NUW8 1/20 0.58
KDM4E B2RXH2 1/20 0.58
F7 P08709 1/20 0.57
F3 P13726 1/20 0.57
SARM1 Q6SZW1 1/20 0.57
SIRT2 Q8IXJ6 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nicotinyl Methylamide SCHEMBL28560459 1.00 HDAC1 (0.69) HDAC1HDAC6MKNK1MKNK2LMNA
Nicotinyl Methylamide SCHEMBL30664356 1.00 HDAC1 (0.69) HDAC1HDAC6MKNK1MKNK2LMNA
Nicotinyl Methylamide SCHEMBL29082835 0.98 HDAC1 (0.67) HDAC1HDAC6MKNK1MKNK2LMNA
Nicotinyl Methylamide SCHEMBL5891238 0.98 HDAC1 (0.67) HDAC1HDAC6MKNK1MKNK2LMNA
Nicotinyl Methylamide SCHEMBL5528294 0.98 HDAC1 (0.67) HDAC1HDAC6MKNK1MKNK2LMNA
Nicotinyl Methylamide SCHEMBL22190415 0.98 HDAC1 (0.67) HDAC1HDAC6MKNK1MKNK2LMNA
Nicotinyl Methylamide SCHEMBL4730618 0.98 HDAC1 (0.67) HDAC1HDAC6MKNK1MKNK2LMNA
Nicotinyl Methylamide SCHEMBL9275531 0.98 HDAC1 (0.67) HDAC1HDAC6MKNK1MKNK2LMNA
Nicotinyl Methylamide SCHEMBL22190418 0.98 HDAC1 (0.67) HDAC1HDAC6MKNK1MKNK2LMNA
Nicotinyl Methylamide SCHEMBL22190891 0.93 MKNK1 (0.64) HDAC1HDAC6MKNK1MKNK2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2744 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122094660-A Composition in the form of an oil-in-water emulsion 2026-05-26 CN claimed
WO-2026106725-A1 CHLOROPHYLL DERIVATIVES, CAROTENOID DERIVATIVES, AND DIETARY SUPPLEMENTS FOR HUMAN OCULAR HEALTH AND VISUAL PERFORMANCE RETINABIO, INC. (US) 2026-05-21 WO claimed
EP-3869192-B1 METHOD FOR QUANTITATIVE DETECTION OF VARIOUS METABOLITES IN BIOLOGICAL SAMPLE HUMAN METABOLOMICS INST INC (CN) 2026-05-13 EP claimed
US-20260076956-A1 METHODS FOR REGRESSING OR REVERSING FIBROSIS AND/OR LIVER CIRRHOSIS IN A SUBJECT IN NEED THEREOF USING HIGH-DOSE NIACIN, OR A NIACIN ANALOG THEREOF US GOV VETERANS AFFAIRS (US) 2026-03-19 US claimed
EP-4687829-A1 COMPOSITION FOR CARING FOR KERATIN MATERIALS L'OREAL (FR) 2026-02-11 EP claimed
EP-4679085-A1 BIOMARKER AND USE THEREOF MEIJI CO., LTD (JP) 2026-01-14 EP claimed
US-20250381116-A1 SOLUBILIZATION OF THIOPYRIDINONE COMPOUND AND COMPOSITION COMPRISING SAME OREAL (FR) 2025-12-18 US claimed
EP-4604968-A1 ENHANCED NAD+ COMPOSITIONS AND METHODS OF MAKING AND USING THE SAME Bionadrx Holdings, Inc. (US) 2025-08-27 EP claimed
US-20250258146-A1 QUANTITATIVE DETECTION METHOD OF MULTIPLE METABOLITES IN BIOLOGICAL SAMPLE AND METABOLIC CHIP HUMAN METABOLOMICS INSTITUTE INC. (CN) 2025-08-14 US claimed
EP-4580589-A1 USE OF A COMPOSITION FOR BOOSTING SKIN'S NIGHT REPAIR ASSOCIATED FUNCTIONS Unilever IP Holdings B.V. (NL) 2025-07-09 EP claimed
WO-1998033786-A9 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS 1998-12-30 WO claimed
WO-1998033786-A1 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS THE SCRIPPS RESEARCH INSTITUTE (US) 1998-08-06 WO claimed
WO-1996020010-A1 COMBINATION FOR REDUCING ANTIMICROBIAL RESISTANCE USING A METHYLATION INHIBITOR IN COMBINATION WITH AN ANTIBIOTIC ORIDIGM CORPORATION (US) 1996-07-04 WO claimed
EP-0527186-A4 UNIV ILLINOIS (US) 1995-01-18 EP claimed
US-5286721-A Antimicrobial agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-02-15 US claimed
EP-0527186-A1 PHOTODYNAMIC PLANT DEFOLIANTS AND CHLOROPHYLL BIOSYNTHESIS MODULATORS The Board of Trustees for the University of Illinois (US) 1993-02-17 EP claimed
EP-0506982-A1 1-AZABICYCLO 3.2.0]HEPT-2-ENE-2-CARBOXYLIC ACID COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-10-07 EP claimed
WO-1992006978-A1 1-AZABICYCLO[3.2.0]HEPT-2-ENE-2-CARBOXYLIC ACID COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-04-30 WO claimed
EP-0303227-B1 ETHERS AND THIOETHERS HAVING THERAPEUTICAL ACTIVITY, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1992-02-05 EP claimed
WO-1991016820-A1 PHOTODYNAMIC PLANT DEFOLIANTS AND CHLOROPHYLL BIOSYNTHESIS MODULATORS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 1991-11-14 WO claimed