SCHEMBL12952016

SCHEMBL12952016

C/C=C(/CN)N1CCn2c(nc(-c3ccc(F)cc3)c2NC2CCCCC2)C1(C)C

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.56
CYP3A4 P08684 1/20 0.56
ALOX5 P09917 5/20 0.43
ADORA1 P30542 2/20 0.35
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
CSNK1E P49674 1/20 0.34
MAPK14 Q16539 4/20 0.34
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TLR9 Q9NR96 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1046633 0.88 KCNH2 (0.72) KCNH2CYP3A4ALOX5ADORA1CSNK1E
SCHEMBL1051312 0.88 KCNH2 (0.72) KCNH2CYP3A4ALOX5ADORA1CSNK1E
SCHEMBL998581 0.87 KCNH2 (0.73) KCNH2CYP3A4ALOX5ADORA1ADORA3
SCHEMBL1049778 0.85 KCNH2 (0.73) KCNH2CYP3A4ALOX5CSNK1E
SCHEMBL15760182 0.81 KCNH2 (0.55) KCNH2CYP3A4
SCHEMBL1051930 0.80 KCNH2 (0.70) KCNH2CYP3A4ALOX5CSNK1E
SCHEMBL1048320 0.80 KCNH2 (0.70) KCNH2CYP3A4MAPK14
SCHEMBL1050854 0.78 KCNH2 (0.68) KCNH2CYP3A4ALOX5CSNK1E
SCHEMBL1048483 0.78 KCNH2 (0.68) KCNH2CYP3A4ALOX5TLR9
SCHEMBL1051385 0.78 KCNH2 (0.70) KCNH2CYP3A4ALOX5MAPK14LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006143-A2 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES IRM LLC (BM) 2011-01-13 WO disclosed