SCHEMBL12952249

SCHEMBL12952249

CC(=O)NCCCCCC(=O)N1CCn2c(nc(-c3ccc(F)cc3)c2Nc2ccc(C)cc2)C1

nearest known ligand 0.71

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.71
CYP3A4 P08684 1/20 0.44
TGFBR1 P36897 2/20 0.36
CSNK1D P48730 2/20 0.36
CSNK1E P49674 2/20 0.36
USP2 O75604 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
NAMPT P43490 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12952259 0.92 KCNH2 (0.69) KCNH2CYP3A4CSNK1DCSNK1EUSP2
SCHEMBL12952247 0.91 KCNH2 (0.68) KCNH2CYP3A4TGFBR1CSNK1DCSNK1E
SCHEMBL2068616 0.91 KCNH2 (0.70) KCNH2CYP3A4TGFBR1CSNK1DCSNK1E
SCHEMBL12952020 0.89 KCNH2 (0.77) KCNH2CYP3A4TGFBR1CSNK1DCSNK1E
SCHEMBL12952026 0.88 KCNH2 (0.78) KCNH2CYP3A4TGFBR1CSNK1DCSNK1E
SCHEMBL20121553 0.87 KCNH2 (0.71) KCNH2CYP3A4TGFBR1CSNK1DCSNK1E
SCHEMBL2069249 0.86 KCNH2 (0.81) KCNH2CYP3A4TGFBR1CSNK1DCSNK1E
SCHEMBL2069854 0.86 KCNH2 (0.65) KCNH2CYP3A4TGFBR1CSNK1DCSNK1E
SCHEMBL12952260 0.86 KCNH2 (0.75) KCNH2CYP3A4TGFBR1CSNK1DCSNK1E
SCHEMBL15750603 0.85 KCNH2 (0.61) KCNH2CYP3A4USP2LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed
WO-2011006143-A2 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES IRM LLC (BM) 2011-01-13 WO disclosed