SCHEMBL12973576

SCHEMBL12973576

CCOC(=O)C1(c2ccc(Oc3ccc(-c4onc(C)c4NC(=O)OC(C)c4ccccc4)cc3)cc2)CC1

nearest known ligand 0.74

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 18/20 0.74
ABCC3 O15438 1/20 0.74
ABCC4 O15439 1/20 0.74
ABCB11 O95342 1/20 0.74
CYP2C8 P10632 1/20 0.74
CYP2C9 P11712 1/20 0.74
ABCB4 P21439 1/20 0.74
ABCC2 Q92887 1/20 0.74
SLCO1B3 Q9NPD5 1/20 0.74
SLCO1B1 Q9Y6L6 1/20 0.74
LPAR3 Q9UBY5 12/20 0.64
LPAR2 Q9HBW0 2/20 0.48
HRH1 P35367 1/20 0.46
KCNA3 P22001 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2761466 1.00 LPAR1 (0.74) LPAR1ABCC3ABCC4ABCB11CYP2C8
SCHEMBL1325246 0.95 LPAR1 (0.82) LPAR1ABCC3ABCC4ABCB11CYP2C8
SCHEMBL8006 0.95 LPAR1 (0.82) LPAR1ABCC3ABCC4ABCB11CYP2C8
SCHEMBL8005 0.95 LPAR1 (0.82) LPAR1ABCC3ABCC4ABCB11CYP2C8
SCHEMBL342934 0.93 LPAR1 (0.78) LPAR1ABCC3ABCC4ABCB11CYP2C8
SCHEMBL342933 0.93 LPAR1 (0.78) LPAR1ABCC3ABCC4ABCB11CYP2C8
SCHEMBL343676 0.92 LPAR1 (0.77) LPAR1ABCC3ABCC4ABCB11CYP2C8
SCHEMBL343677 0.92 LPAR1 (0.77) LPAR1ABCC3ABCC4ABCB11CYP2C8
SCHEMBL2761567 0.91 LPAR1 (0.90) LPAR1ABCC3ABCC4ABCB11CYP2C8
SCHEMBL12973623 0.91 LPAR1 (0.90) LPAR1ABCC3ABCC4ABCB11CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141768-A2 POLYCYCLIC ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-12-09 WO disclosed