SCHEMBL13009508

SCHEMBL13009508

C=C(Nc1ccc(C)c(-c2ccc(C(=O)NCC3CC3)cn2)c1)c1ccoc1

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 20/20 0.64
HSPB1 P04792 2/20 0.64
CYP2C9 P11712 1/20 0.59
MAPK13 O15264 1/20 0.49
MAPK12 P53778 1/20 0.49
MAPK11 Q15759 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3408656 0.92 MAPK14 (0.75) MAPK14HSPB1CYP2C9MAPK13MAPK12
SCHEMBL3404864 0.80 MAPK14 (0.87) MAPK14HSPB1CYP2C9MAPK11
Gw743024X SCHEMBL4817886 0.78 MAPK14 (1.00) MAPK14HSPB1
SCHEMBL3402871 0.78 MAPK14 (0.75) MAPK14HSPB1CYP2C9MAPK13MAPK12
SCHEMBL3406048 0.76 MAPK14 (0.80) MAPK14HSPB1CYP2C9MAPK13MAPK12
SCHEMBL3405640 0.75 MAPK14 (0.68) MAPK14HSPB1CYP2C9MAPK13MAPK12
SCHEMBL3405481 0.75 MAPK14 (1.00) MAPK14HSPB1CYP2C9MAPK11
SCHEMBL14365176 0.75 MAPK14 (0.71) MAPK14HSPB1CYP2C9MAPK11
SCHEMBL14403203 0.75 MAPK14 (0.62) MAPK14CYP2C9MAPK11
SCHEMBL3409280 0.73 P4HTM (0.53) MAPK14HSPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2258687-A1 Nicotinamide derivates useful as P38 inhibitors Glaxosmithkline LLC (US) 2010-12-08 EP disclosed