SCHEMBL13017686

SCHEMBL13017686

OC(CNCCCc1ccccc1)c1cc(C(F)(F)F)nc2c(C(F)(F)F)cccc12

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.76
CYP3A4 P08684 4/20 0.62
CYP2D6 P10635 3/20 0.55
ADORA2A P29274 5/20 0.46
ADORA1 P30542 5/20 0.46
ADORA3 P0DMS8 3/20 0.46
GLRA1 P23415 2/20 0.46
SLC6A2 P23975 2/20 0.46
AVPR2 P30518 2/20 0.46
SLC6A4 P31645 2/20 0.46
HRH1 P35367 2/20 0.46
OPRM1 P35372 2/20 0.46
DRD3 P35462 2/20 0.46
MC3R P41968 2/20 0.46
HTT P42858 2/20 0.46
SLC6A3 Q01959 2/20 0.46
GHSR Q92847 2/20 0.46
ADORA2B P29275 1/20 0.46
CYP2C19 P33261 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18343536 0.94 KCNH2 (0.73) KCNH2CYP3A4CYP2D6ADORA2AADORA1
SCHEMBL18343569 0.89 KCNH2 (0.71) KCNH2CYP3A4CYP2D6ADORA2AADORA1
SCHEMBL11904508 0.88 KCNH2 (0.69) KCNH2CYP3A4CYP2D6ADORA2AADORA1
SCHEMBL11904381 0.88 KCNH2 (0.69) KCNH2CYP3A4CYP2D6ADORA2AADORA1
SCHEMBL7208062 0.88 KCNH2 (0.69) KCNH2CYP3A4CYP2D6ADORA2AADORA1
SCHEMBL12702439 0.88 KCNH2 (0.94) KCNH2CYP3A4CYP2D6ADORA2AADORA1
SCHEMBL11904847 0.87 KCNH2 (1.00) KCNH2CYP3A4CYP2D6ADORA2AADORA1
SCHEMBL11904428 0.87 KCNH2 (1.00) KCNH2CYP3A4CYP2D6ADORA2AADORA1
SCHEMBL12472251 0.87 KCNH2 (1.00) KCNH2CYP3A4CYP2D6ADORA2AADORA1
SCHEMBL12473159 0.86 KCNH2 (1.00) KCNH2CYP3A4CYP2D6ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010144101-A1 NEXT GENERATION QUINOLOINE METHANOLS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY OF THE ARMY, ON BEHALF OF U.S. (US) 2010-12-16 WO disclosed
WO-2010144102-A1 PENTAFLUOROSULFANYL ANALOGS OF MEFLOQUINE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY OF THE ARMY, ON BEHALF OF U.S. ARMY MEDICAL RESEARCH AND MATERIAL COMMAND (US) 2010-12-16 WO disclosed