SCHEMBL13018992

SCHEMBL13018992

CC(=O)OC(OCc1ccccc1)C(C)NC(=O)[C@@H]1CCCCN1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSC P53634 4/20 0.47
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
HTR2C P28335 1/20 0.46
HTR2B P41595 1/20 0.46
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
CTSK P43235 1/20 0.40
KCNH2 Q12809 1/20 0.40
MASP2 O00187 1/20 0.39
GPR88 Q9GZN0 1/20 0.38
SLC6A3 Q01959 2/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
DHFR P00374 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13019452 0.87 CTSC (0.47) CTSCCYP3A4CYP2D6CYP2C9TSHR
SCHEMBL3676422 0.80 HTR2C (0.45) CTSCCYP3A4CYP2D6CYP2C9TSHR
SCHEMBL14131110 0.78 HTR2C (0.54) CTSCCYP3A4CYP2D6CYP2C9TSHR
Hydrochloric Acid SCHEMBL5095147 0.78 HTR2C (0.53) CTSCCYP3A4CYP2D6CYP2C9TSHR
SCHEMBL10934562 0.78 CTSC (0.55) CTSCCYP3A4CYP2D6CYP2C9TSHR
SCHEMBL31364184 0.75 CTSC (0.53) CTSCCYP3A4CYP2D6CYP2C9TSHR
SCHEMBL8130551 0.75 HTR2C (0.57) CTSCCYP3A4CYP2D6CYP2C9TSHR
SCHEMBL9115117 0.75 HTR2C (0.57) CTSCCYP3A4CYP2D6CYP2C9TSHR
SCHEMBL8773336 0.75 HTR2C (0.57) CTSCCYP3A4CYP2D6CYP2C9TSHR
SCHEMBL8130548 0.75 HTR2C (0.57) CTSCCYP3A4CYP2D6CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2261232-A2 Inhibitors of caspases VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-12-15 EP disclosed