SCHEMBL13043314

SCHEMBL13043314

O=C(Nc1cccc(Nc2c(N3CCCCC3)c(=O)c2=O)c1)c1sccc1NCc1ccnc2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.53
RET P07949 3/20 0.53
KIT P10721 2/20 0.53
RAF1 P04049 1/20 0.53
LCK P06239 1/20 0.53
CYP3A4 P08684 1/20 0.53
MAP3K20 Q9NYL2 1/20 0.53
RIPK3 Q9Y572 1/20 0.53
FLT1 P17948 4/20 0.46
P2RX7 Q99572 1/20 0.39
DNMT1 P26358 1/20 0.37
DNMT3A Q9Y6K1 1/20 0.37
FAAH O00519 1/20 0.36
MAPK8 P45983 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK10 P53779 1/20 0.36
AURKA O14965 1/20 0.35
PDPK1 O15530 1/20 0.35
RPS6KB1 P23443 1/20 0.35
AURKB Q96GD4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3731838 0.93 KDR (0.52) KDRRETKITRAF1LCK
SCHEMBL3732453 0.93 KDR (0.59) KDRRETKITRAF1LCK
SCHEMBL3738330 0.93 KDR (0.51) KDRRETKITRAF1LCK
SCHEMBL3735497 0.93 KDR (0.51) KDRRETKITRAF1LCK
SCHEMBL3735473 0.92 KDR (0.51) KDRRETKITRAF1LCK
SCHEMBL13043337 0.91 KDR (0.50) KDRRETKITRAF1LCK
SCHEMBL3748316 0.90 KDR (0.50) KDRRETKITRAF1LCK
SCHEMBL3745989 0.90 KDR (0.48) KDRRETKITRAF1LCK
SCHEMBL3731993 0.89 KDR (0.49) KDRRETKITRAF1LCK
SCHEMBL3735052 0.88 KDR (0.51) KDRRETKITRAF1LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7829717-B2 (Arylamidoaryl)squaramide compounds OSI PHARMACEUTICALS, INC. (US) 2010-11-09 US disclosed
US-7829717-B2 (Arylamidoaryl)squaramide compounds OSI PHARMACEUTICALS, INC. (US) 2010-11-09 US disclosed