SCHEMBL13070517

SCHEMBL13070517

CCc1c2n(c(=O)c3c(OC)c(OC)ccc13)CCc1cc(O)c(O)cc1-2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.44
GSK3B P49841 1/20 0.41
CDK5 Q00535 1/20 0.41
CDK5R1 Q15078 1/20 0.41
KDM4E B2RXH2 3/20 0.39
MAPT P10636 3/20 0.39
CYP3A4 P08684 3/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
MEN1 O00255 1/20 0.39
ALOX15 P16050 1/20 0.39
CASP1 P29466 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
RAC1 P63000 2/20 0.39
CYP1B1 Q16678 2/20 0.39
ACHE P22303 1/20 0.38
MAOB P27338 1/20 0.38
KCNK3 O14649 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13071079 0.87 BCHE (0.46) BCHEGSK3BCDK5CDK5R1KDM4E
SCHEMBL299042 0.85 BCHE (0.63) BCHEKDM4EMAPTCYP3A4ALDH1A1
SCHEMBL13070794 0.76 BCHE (0.72) BCHEGSK3BCDK5CDK5R1KDM4E
SCHEMBL31472746 0.75 BCHE (0.65) BCHEKDM4EMAPTCYP3A4ALDH1A1
SCHEMBL31472748 0.75 BCHE (0.65) BCHEKDM4EMAPTCYP3A4ALDH1A1
SCHEMBL31472747 0.75 BCHE (0.65) BCHEKDM4EMAPTCYP3A4ALDH1A1
SCHEMBL18037451 0.74 BCHE (0.58) BCHEKDM4EMAPTCYP3A4ALDH1A1
SCHEMBL299656 0.74 BCHE (0.58) BCHEKDM4EMAPTCYP3A4ALDH1A1
SCHEMBL18037466 0.73 BCHE (0.48) BCHEKDM4EMAPTCYP3A4ALDH1A1
SCHEMBL18037443 0.73 BCHE (0.56) BCHEKDM4EMAPTCYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010128061-A1 NOVEL ISOQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-11-11 WO disclosed