SCHEMBL13075337

SCHEMBL13075337

COc1cc2c(cc1O)c(=O)[nH]c1c3cc(O)c(O)cc3ncc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 2/20 0.39
CYP1B1 Q16678 2/20 0.39
SRC P12931 1/20 0.39
GUSB P08236 1/20 0.39
CYP1A2 P05177 1/20 0.39
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
EGFR P00533 2/20 0.36
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PDE10A Q9Y233 1/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
RAD52 P43351 1/20 0.35
KMT2A Q03164 1/20 0.35
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL298221 0.71 PARP1 (0.51) SRCEGFRALDH1A1SMN1; SMN2PDPK1
SCHEMBL20967693 0.70 JAK1 (0.54)
SCHEMBL17546677 0.70 MAOB (0.50) KDM4EALDH1A1HPGDMEN1POLB
SCHEMBL8840857 0.70 MAOB (0.50) KDM4EALDH1A1HPGDMEN1POLB
SCHEMBL27041249 0.70 KDM4E (0.56) CYP1A1CYP1B1GUSBCYP1A2PDE3B
SCHEMBL17133045 0.68 MAOB (0.52) KDM4EALDH1A1HPGDMEN1POLB
SCHEMBL8840801 0.68 MAOB (0.52) KDM4EALDH1A1HPGDMEN1POLB
SCHEMBL641721 0.68 SRC (0.54) SRCEGFRALDH1A1SMN1; SMN2PDPK1
SCHEMBL13075718 0.67 TDP1 (0.59) SRCSMN1; SMN2
SCHEMBL20327078 0.67 KDM4E (0.56) CYP1A1CYP1B1GUSBCYP1A2PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127363-A1 TOPOSIOMERASE INHIBITORS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2010-11-04 WO disclosed