SCHEMBL13076282

SCHEMBL13076282

Cc1nn(C)c(C)c1-c1cc(C(=O)c2nc3ccc(OC4CCN(C)CC4)nc3[nH]2)ccc1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 2/20 0.43
CCND1 P24385 2/20 0.43
CCND3 P30281 1/20 0.43
CDK6 Q00534 1/20 0.43
JAK3 P52333 1/20 0.40
CHEK2 O96017 2/20 0.38
BRD4 O60885 1/20 0.33
LCK P06239 1/20 0.33
KDR P35968 1/20 0.33
MAPK14 Q16539 1/20 0.33
MAP4K1 Q92918 1/20 0.33
HRH4 Q9H3N8 2/20 0.32
SCN1A P35498 1/20 0.32
SCN2A Q99250 1/20 0.32
SCN3A Q9NY46 1/20 0.32
FPR2 P25090 1/20 0.32
PROKR1 Q8TCW9 1/20 0.32
MAPK7 Q13164 1/20 0.32
ATR Q13535 1/20 0.31
GSK3B P49841 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL112968 0.79 CDK4 (0.52) CDK4CCND1CCND3CDK6JAK3
SCHEMBL13075594 0.75 CDK4 (0.43) CDK4CCND1CCND3CDK6
SCHEMBL111269 0.74 CDK4 (0.49) CDK4CCND1CCND3CDK6
SCHEMBL112506 0.71 CDK4 (0.63) CDK4CCND1CCND3CDK6
SCHEMBL110403 0.70 CDK4 (0.62) CDK4CCND1CCND3CDK6ATR
SCHEMBL111573 0.69 CDK4 (0.80) CDK4CCND1CCND3CDK6
SCHEMBL111484 0.68 CDK4 (0.62) CDK4CCND1CCND3CDK6
SCHEMBL2143455 0.68 CDK4 (0.51) CDK4CCND1CCND3CDK6
SCHEMBL13076251 0.66 CDK4 (0.48) CDK4CCND1CCND3CDK6ATR
SCHEMBL112177 0.64 CDK4 (0.75) CDK4CCND1CCND3CDK6MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125402-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS MODULATORS OF CYCLIN DEPENDENT KINASES NOVARTIS AG (CH) 2010-11-04 WO disclosed