SCHEMBL13076353

SCHEMBL13076353

C=C(C)Nc1ccc(Cl)nc1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 17/20 0.51
KCNQ2 O43526 17/20 0.51
KCNE1 P15382 12/20 0.51
KCNQ1 P51787 12/20 0.51
BACE1 P56817 1/20 0.50
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
ALDH1A1 P00352 1/20 0.43
TNF P01375 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL203109 0.82 KCNQ3 (0.54) KCNQ3KCNQ2KCNE1KCNQ1BACE1
SCHEMBL5629234 0.81 KCNQ3 (0.60) KCNQ3KCNQ2KCNE1KCNQ1BACE1
SCHEMBL21392142 0.78 NPSR1 (0.47) KCNQ3KCNQ2RAB9ASMN1; SMN2ALDH1A1
SCHEMBL5629229 0.77 KCNQ3 (0.60) KCNQ3KCNQ2KCNE1KCNQ1BACE1
SCHEMBL30568974 0.76 KCNQ3 (0.64) KCNQ3KCNQ2KCNE1KCNQ1BACE1
SCHEMBL6361424 0.76 KCNQ3 (0.64) KCNQ3KCNQ2KCNE1KCNQ1BACE1
SCHEMBL28603489 0.74 KCNQ3 (0.57) KCNQ3KCNQ2KCNE1KCNQ1BACE1
SCHEMBL2436172 0.74 KCNQ3 (0.67) KCNQ3KCNQ2KCNE1KCNQ1BACE1
SCHEMBL7764259 0.74 KCNQ3 (0.49) KCNQ3KCNQ2KCNE1KCNQ1BACE1
SCHEMBL23177712 0.74 KCNQ3 (0.68) KCNQ3KCNQ2KCNE1KCNQ1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010130034-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-11-18 WO disclosed