SCHEMBL13078074

SCHEMBL13078074

CCc1cc(-c2nn[nH]c2-c2ccc(O)cc2)cc(CC)c1CC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 1/20 0.39
ESR1 P03372 5/20 0.37
ESR2 Q92731 5/20 0.37
TNIK Q9UKE5 3/20 0.37
ESRRB O95718 1/20 0.36
ESRRA P11474 1/20 0.36
CCNB2 O95067 1/20 0.34
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
CCNB3 Q8WWL7 1/20 0.34
FGFR1 P11362 1/20 0.34
USP7 Q93009 5/20 0.33
CA12 O43570 1/20 0.33
ALPL P05186 1/20 0.33
RPS6KA3 P51812 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL412079 0.87 TNIK (0.36) TNIK
SCHEMBL409864 0.85 TLR9 (0.39) GSK3B
SCHEMBL412468 0.85 KMT2A (0.43) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL412583 0.84 LRRK2 (0.36)
SCHEMBL13078075 0.84
SCHEMBL409866 0.84 PSMB5 (0.36) GSK3B
SCHEMBL13077869 0.83 ESR1 (0.43) HSD17B1ESR1ESR2TNIKFGFR1
SCHEMBL412348 0.82 MEN1 (0.43) MEN1KMT2A
SCHEMBL411522 0.80 CYP1A2 (0.39)
SCHEMBL412946 0.80 TLR8 (0.42) GSK3AGSK3BCDK5FGFR1RPS6KA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100279410-A1 COMPOUNDS FOR THE TREATMENT OF PROLIFERATIVE DISORDERS SYNTA PHARMACEUTICALS CORP. 2010-11-04 US disclosed