SCHEMBL13080705

SCHEMBL13080705

CC(C)C[C@@H](O)C(=O)N1CCN(c2nc(-c3ccccc3Cl)nc3ccccc23)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.61
MEN1 O00255 4/20 0.59
KMT2A Q03164 4/20 0.59
CYP1A2 P05177 5/20 0.55
CYP3A4 P08684 5/20 0.55
MAPT P10636 4/20 0.55
CYP2D6 P10635 4/20 0.55
HSD17B10 Q99714 2/20 0.55
CYP2C19 P33261 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
SMAD3 P84022 1/20 0.47
ALDH1A1 P00352 3/20 0.47
TSHR P16473 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
GBA1 P04062 3/20 0.46
SMO Q99835 1/20 0.45
HIF1A Q16665 2/20 0.44
AKT1 P31749 1/20 0.44
AKT2 P31751 1/20 0.44
AKT3 Q9Y243 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1624037 0.89 SMAD3 (0.62) ABCB1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL1624034 0.89 SMAD3 (0.62) ABCB1MEN1KMT2ACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL1622840 0.89 SMAD3 (0.61) ABCB1MEN1KMT2ACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL1622839 0.89 SMAD3 (0.61) ABCB1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL4089554 0.88 ABCB1 (0.65) ABCB1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL1623864 0.88 MEN1 (0.47) ABCB1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL1623861 0.88 MEN1 (0.47) ABCB1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL13080736 0.87 ACP1 (0.57) MEN1KMT2ACYP1A2MAPTHSD17B10
SCHEMBL13080669 0.87 ACP1 (0.57) MEN1KMT2ACYP1A2MAPTHSD17B10
SCHEMBL4097324 0.82 ABCB1 (0.70) ABCB1MEN1KMT2ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8283354-B2 Voltage gated sodium and calcium channel inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-10-09 US disclosed