SCHEMBL13080919

SCHEMBL13080919

O=C(NC(Cc1ccc2[nH]c(=O)oc2c1)C(=O)N1CCC(N2CCCCC2)CC1)N1CCC(N2Cc3ccccc3NC2=O)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 19/20 1.00
CYP3A4 P08684 17/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30231948 1.00 CALCRL (1.00) CALCRLCYP3A4
SCHEMBL3605793 1.00 CALCRL (1.00) CALCRLCYP3A4
SCHEMBL3761596 0.96 CALCRL (0.93) CALCRLCYP3A4
SCHEMBL30231332 0.96 CALCRL (0.92) CALCRLCYP3A4
SCHEMBL13081485 0.96 CALCRL (0.92) CALCRLCYP3A4
SCHEMBL3757333 0.96 CALCRL (0.92) CALCRLCYP3A4
SCHEMBL3753943 0.92 CALCRL (0.84) CALCRLCYP3A4
SCHEMBL3760943 0.90 CALCRL (0.81) CALCRLCYP3A4
SCHEMBL14280629 0.90 CALCRL (0.81) CALCRLCYP3A4
SCHEMBL30231479 0.90 CALCRL (0.81) CALCRLCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7842808-B2 calcitonin gene-related peptide receptors antagonists such as 4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperidine-1-carboxylic acid[2-(1,4-dioxa-8-aza-spiro [4.5]dec-8-yl)-1-(1H-indol-5-ylmethyl)-2-oxo-ethyl]-amide, used for treating headaches, pain, hot flashes or respiratory system disorders BRISTOL-MYERS SQUIBB COMPANY (US) 2010-11-30 US disclosed
US-7220862-B2 Calcitonin gene related peptide receptor antagonists BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-22 US disclosed