SCHEMBL13080974

SCHEMBL13080974

O=CC(Cc1ccc2c(c1)CC(=O)N2)NC(=O)N1CCC(N2Cc3ccccc3NC2=O)CC1

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 18/20 0.71
CYP3A4 P08684 8/20 0.71
CALCA P06881 1/20 0.53
CHRM4 P08173 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13283564 0.89 CALCRL (0.76) CALCRLCYP3A4CALCA
SCHEMBL13081132 0.86 CALCRL (0.58) CALCRLCYP3A4CALCA
SCHEMBL3607821 0.85 CALCRL (0.76) CALCRLCYP3A4CALCA
SCHEMBL3607815 0.85 CALCRL (0.76) CALCRLCYP3A4CALCA
SCHEMBL13080975 0.83 CALCRL (0.72) CALCRLCYP3A4CALCA
SCHEMBL27626928 0.83 CALCRL (0.65) CALCRLCYP3A4CALCACHRM4
SCHEMBL3590469 0.83 CALCRL (1.00) CALCRLCYP3A4
SCHEMBL13081277 0.83 CALCRL (1.00) CALCRLCYP3A4
SCHEMBL30231739 0.83 CALCRL (1.00) CALCRLCYP3A4
SCHEMBL13080978 0.82 CALCRL (0.65) CALCRLCYP3A4CALCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7842808-B2 calcitonin gene-related peptide receptors antagonists such as 4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperidine-1-carboxylic acid[2-(1,4-dioxa-8-aza-spiro [4.5]dec-8-yl)-1-(1H-indol-5-ylmethyl)-2-oxo-ethyl]-amide, used for treating headaches, pain, hot flashes or respiratory system disorders BRISTOL-MYERS SQUIBB COMPANY (US) 2010-11-30 US disclosed