SCHEMBL13086554

SCHEMBL13086554

CSc1ccc2cc(O)ccc2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 5/20 0.50
ESR1 P03372 4/20 0.50
TTR P02766 1/20 0.44
CYP3A4 P08684 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
HIF1A Q16665 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP1A2 P05177 2/20 0.39
HSD17B14 Q9BPX1 1/20 0.38
PFKFB3 Q16875 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
APP P05067 1/20 0.36
POLB P06746 2/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36
CASP1 P29466 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16573973 0.78 CYP1A2 (0.64) TDP1CYP1A2HSD17B14PDE3BPDE3A
SCHEMBL31428865 0.78 CYP1A2 (0.63) ESR2ESR1TTRCYP1A2POLB
SCHEMBL906951 0.78 CYP1A2 (0.63) ESR2ESR1TTRCYP1A2POLB
SCHEMBL14894660 0.77 BACE1 (0.53) CYP1A2APPPOLBALDH1A1KDM4E
SCHEMBL5188214 0.74 POLB (0.59) CYP1A2PDE3BPDE3APOLBALDH1A1
SCHEMBL16574004 0.73 CYP1A2 (0.47) CYP3A4TSHRHSD17B10CYP1A2APP
SCHEMBL18713743 0.73 TYMS (0.35) TDP1CYP1A2POLBALDH1A1KDM4E
SCHEMBL29522954 0.73 ESR2 (0.59) ESR2ESR1TTRCYP3A4ALOX15
SCHEMBL1060994 0.73 ESR2 (0.59) ESR2ESR1TTRCYP3A4ALOX15
SCHEMBL2817162 0.71 CYP1A2 (0.58) CYP1A2ALDH1A1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100261679-A1 CSF-1R, Inhibitors, Compositions, and Methods of Use NOVARTIS AG (CH) 2010-10-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100261679-A1 CSF-1R, Inhibitors, Compositions, and Methods of Use CSF1R, CSF3R, MSR1 ESR2 630/4885ESR1 1515/4885TTR 2638/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.